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Chemical Structure : SUVN-502
CAS No.: 701205-60-9
Catalog No.: PC-61500Not For Human Use, Lab Use Only.
SUVN-502 (SUVN502, Masupirdine) is a potent, selective, brain penetrant and orally active 5-HT6 receptor antagonist with Ki of 2.04 nM.
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|---|---|---|---|
| 5 mg | $188 | In stock | |
| 10 mg | $298 | In stock | |
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| 50 mg | Get quote | ||
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SUVN-502 (SUVN502, Masupirdine) is a potent, selective, brain penetrant and orally active 5-HT6 receptor antagonist with Ki of 2.04 nM.
SUVN-502 shows high selectivity over 5-HT2A receptor and other 100 target sites.
SUVN-502 produces synergistic effects in extracellular levels of acetylcholine in the ventral hippocampus combined with donepezil and memantine.
SUVN-502 shows potential for treatment of Alzheimer's disease.
| M.Wt | 478.405 | |
| Formula | C21H24BrN3O3S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
1-((2-bromophenyl)sulfonyl)-5-methoxy-3-((4-methylpiperazin-1-yl)methyl)-1H-indole |
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1. Nirogi R, et al. J Med Chem. 2017 Mar 9;60(5):1843-1859.
2. Nirogi R, et al. J Pharm Biomed Anal. 2017 Apr 14;145:423-430.
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