| Cat. No. |
Product Name |
Information |
| PC-72180 |
GSK549
BET BD2 inhibitor
|
GSK549 (GSK-549) is a potent, highly selective, BD2 domain-selective BET inhibitor with pIC50 of 7.8 (BRD4 BD2), 1150-fold selectivity over BD1. |
| PC-35692 |
BRD4 inhibitor Compound V
|
BRD4 inhibitor Compound V is a domain-selective inhibitor of BRD4 with IC50 of 1.8 uM for BRD4 BD1, displays 6- and 16-fold selectivity for BRD4 over BRD2 and BRD3, respectively. |
| PC-35016 |
IBET151-Az
|
IBET151-Az is a IBET151 derivative for PROTAC synthesis.. |
| PC-35015 |
JQ1-Az
|
JQ1-Az is a JQ1 derivative.. |
| PC-43339 |
(R)-(-)-JQ1 Enantiomer
|
(R)-(-)-JQ1 Enantiomer is the stereoisomer of (+)-JQ1, (+)-JQ-1 is a potent, specific BET bromodomain BRD4 inhibitor, but (-)-JQ1 has no activity.. |
| PC-60198 |
Ischemin sodium
|
A cell permeable CBP bromodomain inhibitor with Kd of 19 uM. |
