| Cat. No. |
Product Name |
Information |
| PC-60088 |
FT-671
USP7 inhibitor
|
FT-671 is a novel potent, specific, non-covalent USP7 inhibitor with Kd of 65 nM (USP7 catalytic domain). |
| PC-60087 |
FT-827
USP7 inhibitor
|
FT-827 is a novel potent, specific, covalent USP7 inhibitor with Kd of 7.8 uM (USP7 catalytic domain). |
| PC-60026 |
USP25 and 28 inhibitor AZ-2
USP25/USP28 inhibitor
|
USP25 and 28 inhibitor AZ-2 is a potent, selective, dual USP25/28 inhibitor with IC50 of 0.9/0.9 uM, respectively. |
| PC-60023 |
USP25 and 28 inhibitor AZ-1
USP25/USP28 inhibitor
|
USP25 and 28 inhibitor AZ-1 (AZ1) is a potent, selective, dual USP25/28 inhibitor with IC50 of 0.7/0.6 uM, respectively. |
| PC-60012 |
GNE-6640
USP7 inhibitor
|
GNE-6640 (GNE6640) is a potent, selective and non-covalent USP7 inhibitor with IC50 of 0.75 uM. |
| PC-60003 |
USP7 inhibitor AD-04
USP7 inhibitor
|
USP7 inhibitor AD-04 ((R)-USP-IN-4) is a highly potent, selective, allosteric USP7 inhibitor with IC50 of 6 nM in FP assays, SPR Kd of 2 nM. |
| PC-42241 |
Ubiquitin Isopeptidase-IN-G5
USP5 inhibitor
|
Ubiquitin Isopeptidase-IN-G5 (NSC 144303) is a small molecule inhibitor of ubiquitin-proteasome system by inhibiting the ubiquitin isopeptidases. |
| PC-42231 |
NSC632839
DUBs inhibitor
|
NSC632839 is a small molecule inhibitor of ubiquitin-proteasome system by inhibiting the ubiquitin isopeptidases, inhibits USP2, USP7, and SENP2 with EC50 values of 45 μM, 37 μM, and 9.8 μM, respectively. |
| PC-45498 |
LDN-57444
UCHL1 inhibitor
|
LDN57444 is a potent, reversible, competitive, active site-directed UCHL1 inhibitor with IC50 of 0.88 uM. |
| PC-45341 |
ML-323
USP1 inhibitor
|
ML323 (ML 323) is a potent, selective, reversible inhibitor of the USP1/UAF1 deubiquitinase complex with IC50 of 76 nM. |
| PC-42288 |
ML364
USP2 inhibitor
|
ML364 is a potent, selective and reversible ubiquitin-specific protease USP2 inhibitor with IC50 of 1.1 uM. |
| PC-43555 |
P-50429
USP7/USP47 inhibitor
|
P-50429 (P50429, P 50429) is a potent, selective, covalent deubiquitinase USP7 (EC50=0.42 uM)/USP47 (EC50=1.0 uM) inhibitor with no inhibition for caspase 3, calpain 1, 20S proteasome and a panel of representative USPs. |
