Cat. No. |
Product Name |
Information |
PC-42467 |
CUDC-101
HDAC/EGFR inhibitor
|
CUDC-101 is a potent, multi-targeted HDAC, EGFR and HER2 inhibitor with IC50 of 4.4, 2.4, and 15.7 nM, respectively. |
PC-42468 |
Panobinostat
HDAC inhibitor
|
A potent, broad-spectrum HDAC inhibitor with IC50 of 5-20 nM in cell-free assyas. |
PC-45051 |
Remodelin
|
Remodelin is a potent inhibitor of the acetyl-transferase protein NAT10 that acetylates both histones and microtubules. |
PC-42465 |
Vorinostat
HDAC inhibitor
|
Vorinostat (SAHA) is a potent HDAC inhibitor, inhibits the activities of HDAC1 and HDAC3 with IC50 of 10 nM and 20 nM, respectively. |
PC-42469 |
Belinostat
|
Belinostat (PXD101, PX105684) is a potent HDAC inhibitor with IC50 of 27 nM (HeLa cell extracts). |
PC-45609 |
ACY-738
|
ACY-738 (ACY738) is a potent and specific HDAC6 inhibitor (IC50=1.7 nM) with improved brain bioavailability. |
PC-45583 |
UF-010
class I HDAC inhibitor
|
UF-010 is a potent and selective inhibitor of class I HDACs with IC50s of 0.5/0.1/0.06/1.5/9.1/15.3/44.5 uM for HDAC1/2/3/8/6/10/11 respectively. |
PC-45462 |
TMP-269
class IIa HDAC inhibitor
|
TMP-269 (TMP269) is a potent and selective class IIa HDAC inhibitor with IC50s of 126/80/36/19 nM for HDAC4/5/7/9. |
PC-45089 |
MC-1568
|
MC1568 is a potent and selective class IIa HDAC inhibitor with IC50 of 220 nM for maize HD1-A. |
PC-42902 |
Entinostat
class I HDAC inhibitor
|
Entinostat (MS275) is a potent and selective class I HDACs inhibitor with IC50 of 243/453/248 nM for HDAC1/2/3. |
PC-42671 |
Valproic acid sodium salt
HDAC inhibitor
|
Valproic acid sodium salt is a HDAC inhibitor that selectively inhibits the catalytic activity of class I HDACs, and induces proteasomal degradation of HDAC2. |
PC-42670 |
Valproic acid
HDAC inhibitor
|
Valproic acid is a HDAC inhibitor that selectively inhibits the catalytic activity of class I HDACs, and induces proteasomal degradation of HDAC2. |