| Cat. No. |
Product Name |
Information |
| PC-35321 |
CPTH6 hydrobromide
GCN5/PCAF inhibitor
|
CPTH6 hydrobromide is a thiazole derivative that can reduce histone acetylation and histone acetyltransferase (HAT) activity in human leukemia cells, CPTH6 is a specific Gcn5/pCAF inhibitor. |
| PC-35320 |
CPTH6
GCN5/PCAF inhibitor
|
CPTH6 is a thiazole derivative that can reduce histone acetylation and histone acetyltransferase (HAT) activity in human leukemia cells, CPTH6 is a specific Gcn5/pCAF inhibitor. |
| PC-35191 |
MC2884
HAT/EZH2 inhibitor
|
MC2884 is a novel hybrid, dual HAT/EZH2 inhibitor with IC50 of 3.27, 8.35 and 4.56 uM for CBP, KAT5 and p300, respectively. |
| PC-62558 |
Garcinol
p300/PCAF inhibitor
|
Garcinol (Camboginol) is a potent, natural inhibitor of histone acetyltransferases (HATs) p300 (IC50=7 uM) and PCAF (IC50=5 uM) both in vitro and in vivo. |
| PC-62267 |
SPV106
p300/PCAF activator
|
SPV 106 is the first mixed activator/inhibitor of Histone acetyltransferases (HATs), potentiates p300/CBP-associated factor (PCAF) HAT activity while inhibiting those of p300/CBP and recombinant CBP. |
| PC-62266 |
CTPB
p300 activator
|
CTPB is an anacardic acid derivative, was reported as a selective activator of p300 (KAT3B) HAT activity but not PCAF (KAT2B), which enhanced HAT-dependent transcriptional activation. |
| PC-61762 |
L-002
KAT3B inhibitor
|
L-002 (NSC 764414, L002) is a novel potent, specific acetyltransferase p300 (KAT3B) inhibitor with IC50 of 1.98 uM. |
| PC-61686 |
PU-139
HAT inhibitor
|
PU-139 is a potent, unselective HAT (Histone acetyltransferase) inhibitor that blocks the HATs Gcn5, p300/CBP-associated factor (PCAF), CREB protein (CBP) and p300. |
| PC-61685 |
PU-141
p300/CBP inhibitor
|
PU-141 is a potent, selective CBP/p300 inhibitor that inhibits SK-N-SH cell growth with GI50 of 0.48 uM. |
| PC-60499 |
TH1834 dihydrochloride
Tip60 inhibitor
|
TH1834 dihydrochloride (TH-1834, TH 1834) is a novel potent specific histone acetyltransferase Tip60 inhibitor. |
| PC-60498 |
TH1834
Tip60 inhibitor
|
TH1834 (TH-1834, TH 1834) is a novel potent specific histone acetyltransferase Tip60 inhibitor. |
| PC-70121 |
Windorphen
p300 inhibitor
|
Windorphen is a potent, selective inhibitor of p300 histone acetyltransferase (IC50=4.2 uM). |
