Cat. No. |
Product Name |
Information |
PC-45465 |
UNC-1079
|
The piperidine analog of UNC1021. |
PC-42113 |
MS-049
|
A potent, selective, and cell-active dual inhibitor of PRMT4 and PRMT6 with IC50 of 34±10 nM and 43±7 nM, respectively. |
PC-42272 |
UNC3866
|
A potent, selective PRC1 chromodomains antagonist that binds to CBX4 and CBX7 with Kd of 100 nM. |
PC-42740 |
UNC0224
|
A potent, selective G9a/GLP inhibitor with IC50 of 57 nM and 58 nM CLOT biochemical assays. |
PC-45617 |
WDR5-0103
|
A potent MLL1-WDR5 interaction inhibitor with IC50 of 26.4 nM in competitive binding assay. |
PC-45602 |
MI-136
|
A potent Menin-MLL interaction inhibitor with IC50 of 31 nM. |
PC-44607 |
UNC1215
|
A potent and selective chemical probe for the methyllysine (Kme) reading function of L3MBTL3 with Kd of 120 nM. |
PC-42037 |
HLCL-61 hydrochloride
|
A novel potent and selective protein arginine methyltransferase PRMT5 inhibitor. |
PC-42741 |
UNC0321
|
A highly potent, selective G9a inhibitor with Ki of 63 pM. |
PC-45489 |
PFI-2 hydrochloride
|
A first-in-class, potent and selective inhibitor of SETD7 methyltransferase with Ki app/IC50 of 0.33/2 nM. |
PC-45488 |
PFI-2
|
A first-in-class, potent and selective inhibitor of SETD7 methyltransferase with Ki app/IC50 of 0.33/2 nM. |