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Request The Product List ofAdenosine Receptor Adenosine Receptor

Cat. No. Product Name Information
PC-22013

CVT-6694

A2BR antagonist

CVT-6694 (CVT6694) is a highly potent, selective A2B adenosine receptor antagonist with Ki of 7 nM (hA2B), >700-fold selective over human A1, A2A and A3 receptors.
PC-21513

TRR469

A1AR modulator

TRR469 is a potent, selective adenosine A1 receptor (A1AR) positive allosteric modulator with pKb of 5.36, exhibits anti-nociceptive properties in acute and neuropathic pain models in mice.
PC-21512

VCP171

A1AR modulator

VCP171 is a selective adenosine A1 receptor (A1AR) positive allosteric modulator (PAM), inhibits eEPSC amplitude of nerve-injury versus control animals in both lamina I and lamina II neurons.
PC-21510

MRS7935

A1AR modulator

MRS7935 is a potent, selective positive allosteric modulator (PAM) of A1 adenosine receptor (A1AR) with EC50 of 1.43 uM.
PC-20642

I-ABOPX

A3AR antagonist

I-ABOPX is a potent, selective A3 adenosine receptor antagonist with high affinity for both the ovine (Ki=3 nM) and human (Ki=19 nM) A3 receptors.
PC-20640

QAF-805

A2BR antagonist

QAF-805 (QAF805) is a potent, dual adenosine-A2B receptor and adenosine-A3 receptor antagonist with Ki of 3.4 nM (A2B).
PC-20639

KF26777

A3AR antagonist

KF-26777 (KF26777) is a potent and selective adenosine A3 receptor antagonist with Ki of 0.2 nM (human A3 receptor).
PC-20638

LAS101057

A2BR antagonist

LAS101057 (LAS 101057) is a potent, selective, and orally efficacious A2B adenosine receptor antagonist with Ki of 24 nM (human A2B).
PC-20546

PSB-1115

A2B antagonist

PSB-1115 (PSB1115) is a potent, selective adenosine A2B receptor antagonist with binding Ki of 53.4 nM (recombinant human A2B receptor), 40- and 400-fold selectivity over A1 and A2A receptors.
PC-20111

ASP5854

A1/A2A receptor antagonist

ASP5854 (ASP-5854) is a potent adenosine A(1) and A(2A) receptor dual antagonist with binding Ki of 9.03 and 1.76 nM for human A(1) and A(2A) receptors, respectively.
PC-20110

SCH-442416

A2AR antagonist

SCH-442416 (SCH442416) is a potent, selective and brain-penetrant antagonist of adenosine A2A receptor (A2AR) with Ki 0.048 nM and 0.5 nM for human and rat A2AR, respectively.
PC-20102

KW-6356

A2A receptor antagonist

KW-6356 (Sipagladenant) is a potent and selective adenosine A2A receptor antagonist/inverse agonist with pKi value of9.93 for human A2A receptor.

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