| Cat. No. |
Product Name |
Information |
| PC-49105 |
BnOCPA
|
BnOCPA is a potent and powerful analgesic and a highly selective and potent, full agonist at human adenosine A1 receptors (A1Rs) with pEC50 of 7.23 in a NanoBRET agonist binding assay. |
| PC-35841 |
AB928
|
Etrumadenant (AB928) is a potent, dual antagonist of the A2aR and A2bR adenosine receptors with Kb of 1.5 and 2.0 nM, respectively. |
| PC-35779 |
PBF509
|
PBF509 (Taminadenant, PBF-509, NIR 178) is a novel selective and potent Adenosine A2A Receptor (A2AR) antagonist, antagonizes A2AR agonist-mediated cAMP accumulation and impedance responses with KB values of 72.8 and 8.2 nM, respectively. |
| PC-43007 |
2-Cl-IB-MECA
|
2-Cl-IB-MECA (Chloro-IB-MECA, CF-102, Namodenoson) is a potent, selective A3 adenosine receptor agonist with Ki of 0.33 nM, 2500- and 1400-fold selectivity over A1 and A2a receptors. |
| PC-63144 |
AZD-4635
|
AZD-4635 (HTL 1071) is a potent, selective and orally available adenosine 2A receptor (A2AR) inhibitor with Ki of 1.7 nM, > 30-fold selectivity over other adenosine receptors. |
| PC-70072 |
ST-1535
|
ST1535 is a potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM. |
| PC-20644 |
VUF-5574
|
VUF-5574 (VUF5574) is a potent, selective A3 adenosine receptor antagonist with high affinity (Ki=4.03 nM, human A3 receptor). |
