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Cat. No. Product Name Information
PC-49105

BnOCPA

BnOCPA is a potent and powerful analgesic and a highly selective and potent, full agonist at human adenosine A1 receptors (A1Rs) with pEC50 of 7.23 in a NanoBRET agonist binding assay.
PC-35841

AB928

Etrumadenant (AB928) is a potent, dual antagonist of the A2aR and A2bR adenosine receptors with Kb of 1.5 and 2.0 nM, respectively.
PC-35779

PBF509

PBF509 (Taminadenant, PBF-509, NIR 178) is a novel selective and potent Adenosine A2A Receptor (A2AR) antagonist, antagonizes A2AR agonist-mediated cAMP accumulation and impedance responses with KB values of 72.8 and 8.2 nM, respectively.
PC-43007

2-Cl-IB-MECA

2-Cl-IB-MECA (Chloro-IB-MECA, CF-102, Namodenoson) is a potent, selective A3 adenosine receptor agonist with Ki of 0.33 nM, 2500- and 1400-fold selectivity over A1 and A2a receptors.
PC-63144

AZD-4635

AZD-4635 (HTL 1071) is a potent, selective and orally available adenosine 2A receptor (A2AR) inhibitor with Ki of 1.7 nM, > 30-fold selectivity over other adenosine receptors.
PC-70072

ST-1535

ST1535 is a potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM.
PC-20644

VUF-5574

VUF-5574 (VUF5574) is a potent, selective A3 adenosine receptor antagonist with high affinity (Ki=4.03 nM, human A3 receptor).

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