| Cat. No. |
Product Name |
Information |
| PC-20307 |
BAY-6096
|
BAY-6096 (BAY6096) is a potent, selective, and highly water-soluble adrenergic α2B antagonist with IC50 of 14 nM. |
| PC-49058 |
AS408
|
AS408 is a negative allosteric modulator of the β2-adrenergic receptor (β2AR) for both G-protein activation and arrestin recruitment (pKB=6.8, [35S]GTPγS binding assays), binds to a pocket formed by the membrane-facing surface of TM3 and TM5. |
| PC-47093 |
Tasipimidine
|
Tasipimidine is a potent, selective and orally active human α2A-adrenoceptor agonist with pEC50 of 7.57, >100-fold selectivity over α2B-and α2C-adrenoceptors and the rodent α2D-adrenoceptor. |
| PC-36084 |
Olodaterol hydrochloride
|
Olodaterol hydrochloride (BI1744 CL) is a potent, selective long-acting β2 adrenoceptor agonist with EC50 of 1.4 nM for hβ2. |
| PC-62018 |
BRL 37344 sodium
|
BRL 37344 sodium (BRL 37344A) is a potent and selective β3 adrenoceptor agonist with Ki of 287 nM. |
| PC-62017 |
CL 316243
|
CL 316243 (BTA 243) is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM. |
| PC-62016 |
CL 316243 disodium
|
CL 316243 is a potent, highly selective, orally active β3-adrenoceptor agonist with EC50 of 3 nM. |
