Cat. No. |
Product Name |
Information |
PC-49177 |
BDM88951
|
BDM88951 (BDM 88951) is a highly potent, selective inhibitor of endoplasmic reticulum aminopeptidase 2 (ERAP2) with IC50 of 19 nM. |
PC-72623 |
ST-115
|
ST-115 (ST115) is a potent and specific inhibitor of aminopeptidase P2 ((XPNPEP2, APP2) with IC50 of 3.7 nM. |
PC-35112 |
TP-004
|
TP-004 is a potent, selective and reversible inhibitor of methionine aminopeptidase 2 (MetAP2) with IC50 of 6 nM. |
PC-63317 |
A-832234
|
A-832234 is a potent, selective, reversible MetAP2 inhibitor with IC50 of 19 nM.. |
PC-63184 |
ZGN-1061
|
ZGN-1061 (Aclimostat) is a novel potent, selective Methionine aminopeptidase 2 (MetAP2) inhibitor being investigated for treatment of diabetes and obesity. |
PC-70071 |
Tosedostat
|
Tosedostat (CHR-2797, CHR2797) is a potent, orally bioavailable aminopeptidases inhibitor with IC50 of 150, 220 and 100 nM for PuSA, aminopeptidase N and leucine aminopeptidase, respectively. |
PC-20620 |
Actinonin
|
Actinonin is an isolated antibiotic and shown to be an inhibitor of aminopeptidase M, inhibits enkephalin-degrading enzymes from guinea-pig striatum (enkephalin-aminopeptidase), striatal membrane neutral endopeptidase and soluble dipeptidylaminopeptidase in rat whole brain homogenate with IC50 of 0.39, 5.6 and 1.1 uM, respectively. |