Cat. No. |
Product Name |
Information |
PC-72732 |
DCP1-3
|
DCP1-3 is a novel allosteric ligand of the angiotensin receptor AT1R, displays NAM potency on AngIV with IC50 of 0.29 uM. |
PC-20515 |
Sparsentan
|
Sparsentan (RE-021, DARA-a) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Ki values of 0.8 and 9.3 nM, respectively. |
PC-49657 |
Forasartan
|
Forasartan (SC-52458) is a potent, specific, competitive and reversible angiotensin II receptor (AT1 receptor) antagonist with binding Ki value of 2.9 nM. |
PC-73402 |
Azilsartan mopivabil
|
Azilsartan mopivabil is a potent, selective angiotensin II receptor (AT2R) antagonist, with potential for hypertension, chronic heart failure and diabetic nephropathy. |
PC-73401 |
Azilsartan mepixetil
|
Azilsartan mepixetil is a potent, selective angiotensin II receptor antagonist, with potential for hypertension, chronic heart failure and diabetic nephropathy. |
PC-35877 |
TD-0212
|
TD-0212 (TD0212) is a potent, orally efficacious, dual AT1 antagonist/Neprilysin (NEP) inhibitor with pKi of 8.9 (AT1) and pIC50 of 9.2 (NEP). |
PC-43383 |
EMA401
|
EMA401 (Olodanrigan) is a potent, highly selective angiotensin II type 2 receptor (AT2R) antagonist, inhibits capsaicin responses in cultured neurons of human and rat DRG with IC50 of 10 nM. |