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Cat. No. Product Name Information
PC-72952

BMS-846372

BMS-846372 (BMS846372) is a potent, selective, orally active CGRP receptor antagonist with Ki of 0.07 nM (hCGRP).
PC-38690

Zavegepant

Zavegepant (BHV-3500, BMS-742413)) is a high affinity, selective antagonist of calcitonin gene-related peptide (CGRP) receptor (hCGRP, Ki=0.023 nM), has demonstrated efficacy in the acute treatment of migraine.
PC-72787

FE 205030

FE 205030 (FE205030) is a potent, selective peptidic CGRP antagonist with IC50 of 0.2 nM.
PC-35253

Ubrogepant

Ubrogepant (MK-1602) is a novel potent, selective, oral calcitonin gene-related peptide receptor (CGRP) antagonist for acute treatment of migraine..
PC-62994

MK-8825

MK-8825 is a highly potent, selective, orally bioavailable CGRP receptor antagonist with Ki of 17 nM for rat CGRP.
PC-60031

Atogepant

A potent, selective and orally available CGRP receptor antagonist for the prevention of migraine..
PC-42296

Olcegepant (hydrochloride)

The first small molecule selective CGRP antagonist with Ki of 14.4 nM for hCGRP.

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