Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.

You are here:Home-Chemical Inhibitors & Agonists-Apoptosis-DAPK

Request The Product List ofDAPK DAPK

Cat. No. Product Name Information
PC-38745

CK156

STK17A (DRAK1) inhibitor

CK156 is a potent, highly selective serine/threonine kinase 17A (DRAK1) inhibitor with Kd of 21 nM, cellular IC50 of 182 nM.
PC-38222

SGC-STK17B-1

STK17B (DRAK2) inhibitor

SGC-STK17B-1 is a potent, selective, ATP-competitive inhibitor of death-associated protein kinase family member STK17B (DRAK2) with IC50 of 34 nM, >100-fold selectivity over STK17A.
PC-38221

Dual DRAK1 and DRAK2 inhibitor 1

DRAK2/1 inhibitor

Dual DRAK1 and DRAK2 inhibitor 1 is a potent, dual DRAK2/1 inhibitor Kd value of 9/5 nM, respectively.
PC-35494

HS148

DAPK3 inhibitor

HS148 (DAPK3 inhibitor HS148) is a selective DAPK3 inhibitor with Ki of 119 nM, >10-fold selectivity over Pim kinases..
PC-35493

HS94

DAPK3 inhibitor

HS94 (DAPK3 inhibitor HS94) is a selective DAPK3 inhibitor with Ki of 126 nM, >20-fold selectivity over Pim kinases.
PC-35492

HS56

Pim/DAPK3 inhibitor

HS56 (Pim-DAPK3 inhibitor HS56) is a potent, dual Pim/DAPK3 inhibitor with Ki of 72 nM (Pim-3) and 315 nM (DAPK3), shows micromolar potency toward Pim-1 and Pim-2 (Ki=1.5 and 17 uM).
PC-62870

HS-38

DAPK1/3 inhibitor

HS-38 is a potent and selective DAPK1 and DAPK3 (ZIPK) inhibitor with IC50 of 200 nM for DAPK1 and Kd of 280 nM for ZIPK.
PC-62719

DRAK2-IN-16

DRAK2 inhibitor

DRAK2-IN-116 is a potent, selective DRAK2 inhibitor with IC50 of 3 nM, shows weak inhibition for DRAK1 (IC50=51 nM) and no significant activity against DAPK1/2/3 (IC50>1 uM)..
PC-23345

BLU7482

STK17B inhibitor

BLU7482 is a potent, selective and orally bioavailable inhibitor of serine/threonine kinase 17B (STK17B, DRAK2) with IC50 of 1.0 nM, 45-fold selective over STK17A.
PC-22727

TC-DAPK6

DAPK1/3 inhibitor

TC-DAPK6 is a potent, specific, ATP-competitiveinhibitor of death associated protein kinase (DAPK) with IC50 of 69 and 225 nM for DAPK1 and ZIPK (DAPK3) respectively.
PC-22555

STK17A/B inhibitor 9

STK17A/B inhibitor

STK17A/B inhibitor 9 is a potent and selective, orally active STK17A/B inhibitor with IC50 of 23 nM (STK17A/DRAK1).

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com