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Cat. No. Product Name Information
PC-47098

ASP8062

ASP8062 is a potent, selective GABA B receptor positive allosteric modulator (PAM), positive allosteric modulating activity for human and rat GABAB receptors, exerts analgesic effects in rat model of fibromyalgia.
PC-38319

Zuranolone

Zuranolone (SAGE-217) is an orally active, positive allosteric modulator of the GABAA receptor with EC50 of 375/299 nM (α1β2γ2/α4β3δ).
PC-35483

KRM-II-81

KRM-II-81 is a selective α2/α3 subtype GABAA receptor ligand (positive allosteric modulator) with EC50 of 937 nM for α3β3γ2 GABAAR.
PC-63442

ONO-8590580

ONO-8590580 is a novel potent, selective GABAA α5 negative allosteric modulator, binds to the benzodiazepine binding sites on recombinant human α5-containing GABAA receptors with Ki of 7.9 nM.
PC-62770

MRK-623

MRK-623 is a potent, α2/α3 subunit functionally selectiviie GABAA receptor agonist..
PC-62098

LAU159

LAU159 is a potent, functionally selective positive modulator of α6β3γ2 GABAA receptor..
PC-62089

PF-06372865

PF-06372865 (Darigabat) is a novel potent, α2/3 functionally selective GABAA receptor positive allosteric modulator.

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