| Cat. No. |
Product Name |
Information |
| PC-72725 |
COB-187
|
COB-187 (COB187) is a highly potent and selective inhibitor of GSK-3 with IC50 of 22/11 nM against GSK-3α/GSK-3β. |
| PC-63311 |
BRD0705
|
BRD0705 is a potent, paralog-selective GSK3α inhibitor with IC50 of 66 nM, 8-fold selectivity over GSK3β (IC50=515 nM). |
| PC-63153 |
1-Azakenpaullone
|
1-Azakenpaullone is an analog of kenpaullone and is a potent, selective GSK3β inhibitor with IC50 of 18 nM, weakly inhibits CDK1/cyclin B and CDK5/p25 (IC50=2.0 and 4.2 uM). |
| PC-60431 |
9-ING-41
|
Elraglusib (9-ING-41) is a novel potent, selective GSK-3β inhibitor with IC50 of 0.7 uM. |
| PC-42428 |
CHIR-99021
|
Laduviglusib (CHIR-99021, CT99021) is a potent, specific GSK-3 inhibitor with IC50 of 5 nM and 10 nM for GSK3β and GSK3α, respectively. |
| PC-42628 |
AR-A014418
|
AR-A014418 is a potent, specific ATP-competitive inhibitor of GSK-3β with Ki/IC50 of 38/104 nM. |
| PC-45724 |
Indirubin-3|-monoxime
|
A potent GSK3β inhibitor with IC50 of 22 nM. |
