| Cat. No. |
Product Name |
Information |
| PC-38171 |
GSK8612
|
GSK8612 (GSK-8612) is a highly selective, potent TBK1 inhibitor, inhibits recombinant TBK1 with pIC50 of 6.8 in biochemical functional assays. |
| PC-35769 |
SR12343
|
SR12343 (SR-12343) is a novel NF-κB essential modulator (NEMO)-binding domain (NBD) mimetic for inhibiting IKK/NF-κB activation, inhibits TNF-α-mediated NF-κB activation with IC50 of 11.34 uM in luciferase assays. |
| PC-61282 |
AS602868
|
AS602868 (SPC 839) is a potent, selective and ATP-competitive inhibitor of IKK2 with IC50 of 60 nM and Ki of 20 nM, also interfers directly with FLT3 kinase activation. |
| PC-61066 |
SU-909
|
SU-909 (SU909, IKKα-IN-48) is a potent, selective IKKα inhibitor with Ki of 0.08±0.07 uM, 10-20-fold selectivity over IKKβ (IC50=1.0±0.28 uM). |
| PC-43044 |
WS-3
|
WS3 is a small molecule that can induce proliferation of β cells with EC50 of 74 nM. |
| PC-45916 |
Bay 65-1942
|
Bay 65-1942 (BAY651942) is a potent, selective, ATP-competitive inhibitor of IKKβ kinase with Ki of 2 nM. |
| PC-42418 |
IMD-0354
|
IMD-0354 (IMD0354) is a potent IκB kinase β (IKKbeta) inhibitor, also is a potent inhibitor of glutamine uptake. |
