3-IN-PP1

Chemical Structure : 3-IN-PP1

CAS No.: 2227110-54-3

Catalog No.: PC-26294Not For Human Use, Lab Use Only.

3-IN-PP1 is a highly potent pan-protein kinase D (PKD) inhibitor with IC50 of 108, 94 and 108 nM for PKD1, PKD2 and PKD3 respectively.

Packing	Price	Stock
5 mg	$158	In stock
10 mg	$258	In stock
25 mg	$428	In stock
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100 mg		Get quote

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Biological Activity

3-IN-PP1 is a highly potent pan-protein kinase D (PKD) inhibitor with IC50 of 108, 94 and 108 nM for PKD1, PKD2 and PKD3 respectively.
3-IN-PP1 (0-40 uM) nhibits PKD mediated phosphorylation of cortactin at Ser-298 in HEK293T cells co-transfected with FLAG-PRKD2 and myc-CTTN.

Physicochemical Properties

M.Wt	306.37
Formula	C17H18N6
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	1-(tert-Butyl)-3-(1H-indol-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine

References

1. Gilles P, et al. Eur J Med Chem. 2020 Nov 1;205:112638.

2. Klaas Verschueren, et al. Medchemcomm. 2017 Mar 1;8(3):640-646.

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3-IN-PP1

Biological Activity

Physicochemical Properties

References

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