| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-61254 |
XX-650-23
|
117739-40-9 |
XX-650-23 is a small molecule inhibitor of CREB, blocks CREB/CBP interaction (IC50=3.2 uM) and disrupts CREB-driven gene expression. |
| PC-70246 |
KG-501
|
18228-17-6 |
A small-molecule antagonist of CREB-CBP interaction, inhibits the cAMP-dependent activation of cellular genes via CREB. |
| PC-38619 |
CREB inhibitor 666-15
|
1433286-70-4 |
CREB inhibitor 666-15 is a potent and selective inhibitor of CREB-mediated gene transcription with IC50 of 81 nM, potently inhibits cancer cell growth without harming normal cells. |
| PC-72794 |
Artepillin C
|
72944-19-5 |
Artepillin C (CREB-CRTC2 inhibitor APC) is an inhibitor of CREB/CRTC2 interaction (IC50=24.5 uM), dissociates the CREB/CRTC2 complex, directly binds to CREB with Kd of 3.2 uM). |
| PC-62067 |
NCGC 00067819
|
847163-23-9 |
NCGC 00067819 is a small molecule compound that potentiates CREB signaling with EC50 of 16 nM in the primary screen and 79 nM in the CHO CRE-β-lactamase confirmation assay. |
| PC-61256 |
Naphthol AS-E
|
92-78-4 |
A cell-permeable inhibitor of the KIX-KID interaction and CREB-mediated gene transcription (IC50=2.26 uM). |
