| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-61482 |
TAI-95
|
1438638-83-5 |
TAI-95 (T-1101, TAI 95) is a potent, orally abioavailable Hec1 inhibitor that disrupts Hec1-Nek2 protein interaction wide anti-cancer spectrum (GI50=14.29-73.65 nM, breast cancer cell lines). |
| PC-61480 |
INH154
|
1587705-63-2 |
INH154 is a novel small molecules disrupting Hec1/Nek2 interaction, inhibits HeLa and MDA-MB-468 cancer cells growth with IC50 of 0.20 and 0.12 uM, respectively. |
| PC-42194 |
INH-6
|
1001753-24-7 |
A small molecule inhibitor of Nek2/Hec1 that inhibits cell growth of MB231, MB468, HeLa and K562 cells with IC50 of 1.7, 2.1, 2.4 and 2.5 uM, respectively. |
| PC-61484 |
HCI-2389
|
|
A potent, specific, irreversible NIMA-related Kinase 2 (NEK2) inhibitor with IC50 of 16.65 nM. |
| PC-61483 |
Nek2 inhibitor (R)-21
|
1364269-10-2 |
A potent and selective NIMA-related Kinase 2 (NEK2) inhibitor with IC50 of 22 nM, >200-fold selectivity over Plk1, Mps1, Aurora A and CDK2. |
| PC-61481 |
TAI-1
|
1334921-03-7 |
A potent, small molecule Hec1 inhibitor that disrupts Hec1-Nek2 protein interaction wide anti-cancer spectrum (GI50=13.48 nM K562 cells). |
| PC-61479 |
Nek2 inhibitor 72
|
|
A potent, ATP-competitive and relative selective Nek2 inhibitor with IC50 of 0.27 uM. |
