| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-73412 |
Cudetaxestat
|
1782070-21-6 |
Cudetaxestat (BLD-0409) is a potent, selective autotaxin (NPP2/ATX) inhibitor under investigation for the treatment of NASH. |
| PC-38008 |
CRT0273750
|
1979939-16-6 |
CRT0273750 (IOA-289) is a potent, seletive inhibitor of autotaxin with IC50 of 1 nM. |
| PC-60695 |
Autotaxin inhibitor compound 1
|
1619971-30-0 |
Autotaxin inhibitor compound 1 (Autotaxin-IN-1) is a potent, selective, orally bioavailable inhibitor of autotaxin with IC50 of 2.2 nM in ex vivo human whole blood assay, does not inhibit related proteins ENPP1 and ENPP7. |
| PC-60640 |
GWJ-A-23
|
1351930-95-4 |
GWJ-A-23 (GWJ-23, GWJ23) is a potent, selective autotaxin inhibitor with Ki of 18 nM, an analog of the known ATX inhibitor S32826 and has improved aqueous solubility compared with the parent compound. |
| PC-60639 |
PAT-048
|
1359983-15-5 |
PAT-048 (PAT048) is a potent, selective, noncompetitive autotaxin inhibitor with IC50 of 1.1 nM against the lysoPLD activity of human ATX. |
| PC-60638 |
PAT-505
|
1782070-85-2 |
PAT-505 (PAT 505, PAT505) is a potent, selective, noncompetitive, and orally active autotaxin inhibitor with IC50 of 2.0 nM against the lysoPLD activity of human ATX. |
| PC-60402 |
GLPG-1690
|
1628260-79-6 |
GLPG-1690 (Ziritaxestat, GLPG1690) is a first-in-class, potent, competitive autotaxin inhibitor with Ki/IC50 of 15 nM/131 nM. |
