| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-63128 |
BAY-1816032
|
1891087-61-8 |
BAY-1816032 (BAY1816032) is a highly potent, selective, orally active BUB1 mitotic checkpoint serine/threonine kinase with IC50 of 7 nM, displays excellent selectivity on a panel of 395 kinases. |
| PC-60310 |
GNE-900
|
1200126-26-6 |
GNE-900 (GNE900) is a potent, selective, ATP-competitive, and orally bioavailable Chk1 inhibitor with IC50 of <1 nM. |
| PC-60276 |
GDC-0575
|
1196541-47-5 |
GDC-0575 (ARRY-575, RG-7741) is a potent, selective and orally bioavailable Chk1 inhibitor with IC50 of 1.2 nM. |
| PC-45427 |
Prexasertib
|
1234015-52-1 |
Prexasertib (LY-2606368) is a potent, selective, ATP-competitive inhibitor of CHK1 with Ki of 0.9 nM. |
| PC-42769 |
AZD-7762
|
860352-01-8 |
AZD-7762 (AZD7762) is a potent and selective inhibitor of Chk1/2 with IC50 of 5 nM. |
| PC-45574 |
CCT-245737
|
1489389-18-5 |
CCT-245737 (SRA-737) is a highly potent, selective, ATP-competitive inhibitor of Chk1 with IC50 of 1.3 nM. |
| PC-49284 |
BML-277
|
516480-79-8 |
BML-277 (BML277) is a potent, selective and ATP-competitive inhibitor of Chk2 serine/threonine kinase with IC50 of 15 nM, >1000-fold selectivity over Chk1 and Cdk1/B kinases. |
