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Cat. No. Product Name Information
PC-23653

TRV120027 TFA

AT1R agonist

TRV027 TFA (TRV120027 TFA) is a potent, selective β-arrestin biased ligand / agonist of angiotensin II type 1 receptor (AT1R), competitively antagonizes angiotensin II-stimulated G protein signaling.
PC-23652

TRV027

AT1R agonist

TRV027 (TRV120027) is a potent, selective β-arrestin biased ligand/agonistof angiotensin II type 1 receptor (AT1R), competitively antagonizes angiotensin II-stimulated G protein signaling.
PC-20515

Sparsentan

Dual AT-II and ETA antagonist

Sparsentan (RE-021, DARA-a) is a highly potent dual angiotensin II and endothelin A receptor antagonist with Ki values of 0.8 and 9.3 nM, respectively.
PC-49657

Forasartan

AT1 receptor inhibitor

Forasartan (SC-52458) is a potent, specific, competitive and reversible angiotensin II receptor (AT1 receptor) antagonist with binding Ki value of 2.9 nM.
PC-73402

Azilsartan mopivabil

AT2R antagonist

Azilsartan mopivabil is a potent, selective angiotensin II receptor (AT2R) antagonist, with potential for hypertension, chronic heart failure and diabetic nephropathy.
PC-73401

Azilsartan mepixetil

AT2R antagonist

Azilsartan mepixetil is a potent, selective angiotensin II receptor antagonist, with potential for hypertension, chronic heart failure and diabetic nephropathy.
PC-72732

DCP1-3

AT1R allosteric modulator

DCP1-3 is a novel allosteric ligand of the angiotensin receptor AT1R, displays NAM potency on AngIV with IC50 of 0.29 uM.
PC-35877

TD-0212

AT1/Neprilysin (NEP) inhibitor

TD-0212 (TD0212) is a potent, orally efficacious, dual AT1 antagonist/Neprilysin (NEP) inhibitor with pKi of 8.9 (AT1) and pIC50 of 9.2 (NEP).
PC-43383

EMA401

AT2R inhibitor

EMA401 (Olodanrigan) is a potent, highly selective angiotensin II type 2 receptor (AT2R) antagonist, inhibits capsaicin responses in cultured neurons of human and rat DRG with IC50 of 10 nM.
PC-43020

CGP-42112

AT2 receptor agonist

CGP-42112 (CGP42112A) is a highly potent, selective Angiotensin-II subtype 2 receptor(AT2 receptor) agonist with Ki of 0.24 nM.
PC-43019

Angiotensin 1-7

Angiotensin (1-7) (Ang-(1-7)) is an active heptapeptide of the Renin-angiotensin system (RAS), inhibits purified canine angiotensin converting enzyme (ACE) activity with IC50 of 0.65 uM.
PC-62642

EMA300

AT2 receptor antagonist

EMA300 (PD121981) is a potent, selective small molecule antagonist of angiotensin II type 2 receptor (AT2R) with >1,000-fold selectivity over AT1 receptor.

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