| Cat. No. |
Product Name |
Information |
| PC-43383 |
EMA401
AT2R inhibitor
|
EMA401 (Olodanrigan) is a potent, highly selective angiotensin II type 2 receptor (AT2R) antagonist, inhibits capsaicin responses in cultured neurons of human and rat DRG with IC50 of 10 nM. |
| PC-43020 |
CGP-42112
AT2 receptor agonist
|
CGP-42112 (CGP42112A) is a highly potent, selective Angiotensin-II subtype 2 receptor(AT2 receptor) agonist with Ki of 0.24 nM. |
| PC-43019 |
Angiotensin 1-7
|
Angiotensin (1-7) (Ang-(1-7)) is an active heptapeptide of the Renin-angiotensin system (RAS), inhibits purified canine angiotensin converting enzyme (ACE) activity with IC50 of 0.65 uM. |
| PC-62642 |
EMA300
AT2 receptor antagonist
|
EMA300 (PD121981) is a potent, selective small molecule antagonist of angiotensin II type 2 receptor (AT2R) with >1,000-fold selectivity over AT1 receptor. |
| PC-70201 |
Candesartan
AT1 receptor antagonist
|
Candesartan (CV-11974) is a potent, selective angiotensin II receptor antagonist, inhibits the binding of [125I] angiotensin II to the bovine adrenal cortical membrane and rabbit aortic membrane with IC50 of 112 nM and 28.6 nM, has potent and long-lasting antihypertensive effects. |
| PC-45692 |
BIBS-39
Angiotensin receptor antagonist
|
BIBS-39 (BIBS 39) is a selective nonpeptide angiotensin II receptor antagonist with Ki of 29 nM and 480 nM for AT1 and AT2 respectively. |
| PC-45274 |
Azilsartan medoxomil monopotassium
AT1 receptor antagonist
|
Azilsartan medoxomil monopotassium (TAK-491) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension. |
| PC-45131 |
Olmesartan medoxomil
AT1 receptor antagonist
|
Olmesartan medoxomil (CS-866) is a prodrug of Olmesartan, a potent, selective angiotensin II receptor antagonist. |
| PC-45130 |
Olmesartan
AT1 receptor antagonist
|
Olmesartan (RNH-6270, CS-088) is a potent, selective angiotensin II receptor antagonist, inhibits [125I]angiotensin II binding to bovine adrenal cortical membranes (angiotensin AT1 receptors) with IC50 of 7.7 nM. |
| PC-45306 |
Candesartan cilexetil
AT1 receptor antagonist
|
Candesartan cilexetil (TCV-116) is a potent, selective angiotensin II receptor antagonist, the prodrug of Candesartan. |
| PC-44124 |
Azilsartan
AT1 receptor antagonist
|
Azilsartan (TAK-536) is a specific and potent angiotensin II type 1 receptor (AT1) antagonist with IC50 of 2.6 nM, used in the treatment of adults with essential hypertension. |
| PC-44046 |
Azilsartan medoxomil
AT1 receptor antagonist
|
Azilsartan medoxomil (TAK-491) is a specific and potent angiotensin II type 1 receptor (AT1) antagonist with IC50 of 2.6 nM, used in the treatment of adults with essential hypertension. |
