BIBS-39 |CAS:133085-33-3 Probechem Biochemicals

Chemical Structure : BIBS-39

CAS No.: 133085-33-3

BIBS-39 (BIBS39;BIBS 39)

Catalog No.: PC-45692Not For Human Use, Lab Use Only.

BIBS-39 is a selective nonpeptide angiotensin II receptor antagonist with Ki of 29 nM and 480 nM for AT1 and AT2 respectively.

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10 mg	$288	In stock
25 mg	$560	In stock
50 mg	$728	In stock

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Biological Activity

BIBS-39 is a selective nonpeptide angiotensin II receptor antagonist with Ki of 29 nM and 480 nM for AT1 and AT2 respectively; shows no high affinity for other receptors, shifts the AII concentration-contractile response curves in isolated rabbit aorta with pA2 of 8.14 and a slope of 1.06; shows effective antihypertensives in the model of the renal hypertensive rat.

Physicochemical Properties

M.Wt	524.6533
Formula	C32H36N4O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	DMSO: ≥ 32 mg/mL
Chemical Name/SMILES	[1,1'-Biphenyl]-2-carboxylic acid, 4'-[[2-butyl-6-[[(cyclohexylamino)carbonyl]amino]-1H-benzimidazol-1-yl]methyl]-

References

1. Zhang J, et al. Eur J Pharmacol. 1992 Jul 21;218(1):35-41.

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BIBS-39 (BIBS39;BIBS 39)

Biological Activity

Physicochemical Properties

References

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