GABA Transporter (GAT) (inhibitors, antagonists, agonists)-ProbeChem.com

Request The Product List ofGABA Transporter (GAT) GABA Transporter (GAT)

Cat. No.	Product Name	Information
PC-62933	CI-966 GAT-1 inhibitor	CI-966 (PD 126141) is a potent, selective inhibitor of the GABA transporter GAT-1 with IC50 of 0.26 and 1.2 uM for human and rat GAT-1, respectively.
PC-62932	CI-966 hydrochloride GAT-1 inhibitor	CI-966 hydrochloride is a potent, selective inhibitor of the GABA transporter GAT-1 with IC50 of 0.26 and 1.2 uM for human and rat GAT-1, respectively.
PC-62931	NNC-711 GAT-1 inhibitor	NNC-711 is a potent and selective inhibitor of GABA uptake by GAT-1 with IC50 of 0.04 uM.
PC-62929	NNC 05-2090 hydrochloride GAT2 inhibitor	NNC 05-2090 is a potent selective GABA transporter inhibitor of mGAT2 with Ki of 1.4 uM.
PC-61113	SNAP5114 GABA transport inhibitor	SNAP5114 is a GABA transport inhibitor with IC50 of 5, 21, 388 and 140 uM for hGAT-3, rGAT-2, hGAT-1 and BGT-1, respectively.
PC-42093	SKF-89976A hydrochloride GAT-1 inhibitor	SKF-89976A hydrochloride is a potent, selective and GABA transporter 1 (GAT1) inhibitor with IC50 of 0.13 uM for hGAT1.
PC-24080	Tiagabine hydrochloride GAT1 inhibitor	Tiagabine hydrochloride is an anticonvulsant agent and selective inhibitor of GABA transporter 1 (GAT1) with Ki of 0.1 uM, potently and selectively inhibits GABA reuptake with IC50 of 67, 446 and 182 nM for [3H]GABA uptake in synaptosomes, neurons and glia, respectively.

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