| Cat. No. |
Product Name |
Information |
| PC-62933 |
CI-966
GAT-1 inhibitor
|
CI-966 (PD 126141) is a potent, selective inhibitor of the GABA transporter GAT-1 with IC50 of 0.26 and 1.2 uM for human and rat GAT-1, respectively. |
| PC-62932 |
CI-966 hydrochloride
GAT-1 inhibitor
|
CI-966 hydrochloride is a potent, selective inhibitor of the GABA transporter GAT-1 with IC50 of 0.26 and 1.2 uM for human and rat GAT-1, respectively. |
| PC-62931 |
NNC-711
GAT-1 inhibitor
|
NNC-711 is a potent and selective inhibitor of GABA uptake by GAT-1 with IC50 of 0.04 uM. |
| PC-62929 |
NNC 05-2090 hydrochloride
GAT2 inhibitor
|
NNC 05-2090 is a potent selective GABA transporter inhibitor of mGAT2 with Ki of 1.4 uM. |
| PC-61113 |
SNAP5114
GABA transport inhibitor
|
SNAP5114 is a GABA transport inhibitor with IC50 of 5, 21, 388 and 140 uM for hGAT-3, rGAT-2, hGAT-1 and BGT-1, respectively. |
| PC-42093 |
SKF-89976A hydrochloride
GAT-1 inhibitor
|
SKF-89976A hydrochloride is a potent, selective and GABA transporter 1 (GAT1) inhibitor with IC50 of 0.13 uM for hGAT1. |
