| Cat. No. |
Product Name |
Information |
| PC-60585 |
Compound 101
|
Compound 101 (GRK2 inhibitor 101, Takeda compound 101, Cmpd101) is a novel membrane-permeable, small-molecule inhibitor of GRK2 and GRK3. |
| PC-45591 |
CCG-215022
|
CCG-215022 (CCG215022) is a potent and selective pan GRK (G protein-coupled receptor kinase) inhibitor with IC50 of 0.15/0.38/3.9 uM for GRK2/5/1 respectively. |
| PC-38542 |
Takeda103A
|
Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5. |
| PC-72421 |
GRK6 inhibitor 18
|
GRK6 inhibitor 18 is a potent, and selective GRK6 inhibitor with IC50 of 8 nM. |
| PC-60588 |
CCG 258001
|
A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM. |
| PC-60587 |
CCG 224061
|
A potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 66 nM. |
| PC-60586 |
CCG 258748
|
A potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM. |
