Welcome to Shanghai Probechem Biochemicals Co Ltd !Global Supplier of Chemical Probes, Inhibitors & Agonists.
Chemical Structure : CCG 258748
Catalog No.: PC-60586Not For Human Use, Lab Use Only.
CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.
Bulk size, bulk discount!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.
CCG 258748 displays 30-fold selectivity over GRK5, and no significant inhibitory activity against GRK1, PKA and ROCK1.
| M.Wt | 448.502 | |
| Formula | C24H25FN6O2 | |
| Appearance | Solid | |
| Storage |
|
|
| Solubility |
10 mM in DMSO |
|
1. Bouley R, et al. Mol Pharmacol. 2017 Dec;92(6):707-717.
Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright
