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Chemical Structure : CCG 258748
Catalog No.: PC-60586Not For Human Use, Lab Use Only.
A potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.
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A potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM; displays 30-fold selectivity over GRK5, and no significant inhibitory activity against GRK1, PKA and ROCK1.
| M.Wt | 448.502 | |
| Formula | C24H25FN6O2 | |
| Appearance | Solid | |
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| Solubility |
10 mM in DMSO |
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1. Bouley R, et al. Mol Pharmacol. 2017 Dec;92(6):707-717.
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