CCG 258748 |CAS: 2410997-49-6 Probechem Biochemicals

Chemical Structure : CCG 258748

CCG 258748 (CCG258748;CCG-258748)

Catalog No.: PC-60586Not For Human Use, Lab Use Only.

CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.

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Biological Activity

CCG 258748 is a potent, selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 8 nM.
CCG 258748 displays 30-fold selectivity over GRK5, and no significant inhibitory activity against GRK1, PKA and ROCK1.

Physicochemical Properties

M.Wt	448.502
Formula	C24H25FN6O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	5-((3S,4R)-3-(((1H-indazol-5-yl)oxy)methyl)piperidin-4-yl)-N-((1H-pyrazol-5-yl)methyl)-2-fluorobenzamide

References

1. Bouley R, et al. Mol Pharmacol. 2017 Dec;92(6):707-717.

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CCG 258748 (CCG258748;CCG-258748)

Biological Activity

Physicochemical Properties

References

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