You are here:Home-Chemical Inhibitors & Agonists-GPCR-CGRP Receptor

Request The Product List ofCGRP Receptor CGRP Receptor

Cat. No. Product Name CAS No. Information
PC-38690

Zavegepant

1337918-83-8 Zavegepant (BHV-3500, BMS-742413)) is a high affinity, selective antagonist of calcitonin gene-related peptide (CGRP) receptor (hCGRP, Ki=0.023 nM), has demonstrated efficacy in the acute treatment of migraine.
PC-72952

BMS-846372

1190363-03-1 BMS-846372 (BMS846372) is a potent, selective, orally active CGRP receptor antagonist with Ki of 0.07 nM (hCGRP).
PC-72787

FE 205030

FE 205030 (FE205030) is a potent, selective peptidic CGRP antagonist with IC50 of 0.2 nM.
PC-35253

Ubrogepant

1374248-77-7 Ubrogepant (MK-1602) is a novel potent, selective, oral calcitonin gene-related peptide receptor (CGRP) antagonist for acute treatment of migraine..
PC-62994

MK-8825

1380887-60-4 MK-8825 is a highly potent, selective, orally bioavailable CGRP receptor antagonist with Ki of 17 nM for rat CGRP.
PC-60031

Atogepant

1374248-81-3 A potent, selective and orally available CGRP receptor antagonist for the prevention of migraine..
PC-42296

Olcegepant (hydrochloride)

586368-06-1 The first small molecule selective CGRP antagonist with Ki of 14.4 nM for hCGRP.

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com