Zavegepant (Vazegepant, BHV-3500) | CGRP antagonist

Chemical Structure : Zavegepant

CAS No.: 1337918-83-8

Zavegepant (Vazegepant, BHV-3500, BMS-742413)

Catalog No.: PC-38690Not For Human Use, Lab Use Only.

Zavegepant (Vazegepant, BHV-3500, BMS-742413) is a high affinity, selective antagonist of calcitonin gene-related peptide (CGRP) receptor (hCGRP, Ki=0.023 nM), has demonstrated efficacy in the acute treatment of migraine.

Packing	Price	Stock
5 mg	$198	In stock
10 mg	$298	In stock
25 mg	$488	In stock
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Biological Activity

Zavegepant (Vazegepant, BHV-3500, BMS-742413) is a high affinity, selective antagonist of calcitonin gene-related peptide (CGRP) receptor (hCGRP, Ki=0.023 nM), has demonstrated efficacy in the acute treatment of migraine.

Physicochemical Properties

M.Wt	638.817
Formula	C36H46N8O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-N-(3-(7-methyl-1H-indazol-5-yl)-1-(4-(1-methylpiperidin-4-yl)piperazin-1-yl)-1-oxopropan-2-yl)-4-(2-oxo-1,2-dihydroquinolin-3-yl)piperidine-1-carboxamide

References

1. Stephen E Mercer, et al. Bioorg Med Chem Lett. 2021 Jan 1;31:127624.

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Zavegepant (Vazegepant, BHV-3500, BMS-742413)

Biological Activity

Physicochemical Properties

References

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