| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-38126 |
CCS1477
|
2222941-37-7 |
CCS1477 (Inobrodib) is an orally bioavailable, potent, and selective inhibitor of the p300/CBP bromodomain, binds to p300 and CBP with Kds of 1.3 and 1.7 nM respectively. |
| PC-36166 |
TTK21
|
709676-56-2 |
TTK21 (CBP-p300 activator TTK21) is a small molecule activator of CBP/p300 histone acetyltransferase activity with a maximal effect at a concentration of 275 uM. |
| PC-35580 |
WM-1119
|
2055397-28-7 |
WM-1119 (WM1119) is a highly potent, selective inhibitor of lysine acetyltransferase KAT6A with Kd of 2 nM, shows greate bioavailability and specificity for KAT6A than WM-8014. |
| PC-35579 |
WM-8014
|
2055397-18-5 |
WM-8014 (WM8014) is a highly potent, selective inhibitor of lysine acetyltransferase KAT6A with Kd of 5 nM and IC50 of 8 nM. |
| PC-61762 |
L-002
|
321695-57-2 |
L-002 (NSC 764414, L002) is a novel potent, specific acetyltransferase p300 (KAT3B) inhibitor with IC50 of 1.98 uM. |
| PC-61686 |
PU-139
|
158093-65-3 |
PU-139 is a potent, unselective HAT (Histone acetyltransferase) inhibitor that blocks the HATs Gcn5, p300/CBP-associated factor (PCAF), CREB protein (CBP) and p300. |
| PC-60499 |
TH1834 dihydrochloride
|
2108830-09-5 |
TH1834 dihydrochloride (TH-1834, TH 1834) is a novel potent specific histone acetyltransferase Tip60 inhibitor. |
