| Cat. No. |
Product Name |
Information |
| PC-73089 |
iP300w
p300/CBP inhibitor
|
iP300w (CP-C27) is a potent, selective, orally bioavailable inhibitor of p300/CBP histone acetyltransferases with IC50 of 19 nM (p300), H3K27Ac EC50 of 5 nM, does not inhibit other HATs. |
| PC-72790 |
IMP-1575
HHAT inhibitor
|
IMP-1575 (IMP1575) is a potent, selective Hedgehog acyltransferase (HHAT) inhibitor with Ki/IC50 of 38 nM/0.75 uM (Acyl-cLIP assay). |
| PC-72712 |
ENL YEATS Domain inhibitor 7
ENL YEATS Domain inhibitor
|
ENL YEATS Domain inhibitor 7 is a selective, small molecule inhibitor of ENL YEATS Domain with IC50 of 0.62 uM in inhibiting the ENL-acetyl-H3 interaction. |
| PC-72392 |
PF-9363
KAT6A/6B inhibitor
|
PF-9363 (CTx-648) is a first-in-class, potent and selective KAT6A/6B inhibitor with Ki of 0.41 nM and 1.2 nM for KAT6A and KAT6B, respectively. |
| PC-72364 |
Cholera Toxin B subunit
p300 activator
|
Cholera Toxin B subunit (CTB) is a small molecule activator of p300 HAT enzyme, stimulats the expression of p300. |
| PC-72239 |
CCT077791
PCAF/p300 inhibitor
|
CCT077791 (CCT077791) is a small molecule inhibitor of PCAF and p300 histone acetyltransferase with IC50 of 2.2 uM and IC95 of 35 uM, respectively. |
| PC-72238 |
NU9056
Tip60 (KAT5) inhibitor
|
NU9056 (NU 9056) is a specific Tip60 (KAT5) histone acetyltransferase inhibitor with IC50 of <2 uM. |
| PC-72165 |
CPI-1612
EP300/CBP inhibitor
|
CPI-1612 (CPI 1612) is a highly potent, selective, orally bioavailable EP300/CBP histone acetyltransferase inhibitor with IC50 of 8.1 nM (EP300 HAT SPA). |
| PC-38289 |
WM-3835
KAT7 inhibitor
|
WM-3835 (WM 3835) is a potent, high-specific, cell-permeable inhibitor of MYST acetyltransferase HBO1 (KAT7 or MYST2). |
| PC-38126 |
CCS1477
p300/CBP inhibitor
|
CCS1477 (Inobrodib) is an orally bioavailable, potent, and selective inhibitor of the p300/CBP bromodomain, binds to p300 and CBP with Kds of 1.3 and 1.7 nM respectively. |
| PC-36166 |
TTK21
CBP/p300 activator
|
TTK21 (CBP-p300 activator TTK21) is a small molecule activator of CBP/p300 histone acetyltransferase activity with a maximal effect at a concentration of 275 uM. |
| PC-35580 |
WM-1119
KAT6A inhibitor
|
WM-1119 (WM1119) is a highly potent, selective inhibitor of lysine acetyltransferase KAT6A with Kd of 2 nM, shows greate bioavailability and specificity for KAT6A than WM-8014. |
