Cat. No. |
Product Name |
CAS No. |
Information |
PC-49083 |
Z0933M
|
1561172-42-6 |
Z0933M is a potent S phase kinase-associated protein 1 (Skp1) inhibitor with Kd of 54 nM, potently inhibits Skp1-F-box protein-protein interactions with Ki value of 231 nM in FP-based in vitro competition assays. |
PC-61056 |
VH 298
|
2097381-85-4 |
VH 298 is a potent, specific cell-active VHL E3 ubiquitin ligase inhibitor that inhibits VHL/HIF-α interaction with Kd of 90 nM in ITC assays. |
PC-60125 |
CC-885
|
1010100-07-8 |
CC-885 (CC 885, CC885) is a novel E3 ligase cereblon (CRBN) modulator with potent anti-tumour activity mediated through the degradation of GSPT1. |
PC-60116 |
VH-032
|
1448188-62-2 |
VH-032 (VHL ligand 1) is a VHL ligand for PROTAC and potent, small molecule inhibitor of the VHL/HIF-1α interaction with Kd of 185 nM.. |
PC-60115 |
VHL Ligand 3 (VH032-Boc)
|
1448189-98-7 |
(S,R,S)-AHPC-Boc (VH032-Boc) is a ligand used in the recruitment of the von Hippel-Lindau (VHL) protein and PROTAC technology. |
PC-38766 |
EN106 derivative 3
|
2709040-02-6 |
EN106 derivative 3 is a EN106 derivative used for PROTAC design, EN106 is a covalent ligand and recruiter for FEM1B E3 ligase for targeted protein degradation. |
PC-38765 |
EN106 derivative 2
|
2709040-09-3 |
EN106 derivative 2 is a EN106 derivative used for PROTAC design, EN106 is a covalent ligand and recruiter for FEM1B E3 ligase for targeted protein degradation. |