| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-35841 |
AB928
|
2239273-34-6 |
Etrumadenant (AB928) is a potent, dual antagonist of the A2aR and A2bR adenosine receptors with Kb of 1.5 and 2.0 nM, respectively. |
| PC-35779 |
PBF509
|
1337962-47-6 |
PBF509 (Taminadenant, PBF-509, NIR 178) is a novel selective and potent Adenosine A2A Receptor (A2AR) antagonist, antagonizes A2AR agonist-mediated cAMP accumulation and impedance responses with KB values of 72.8 and 8.2 nM, respectively. |
| PC-43007 |
2-Cl-IB-MECA
|
163042-96-4 |
2-Cl-IB-MECA (Chloro-IB-MECA, CF-102, Namodenoson) is a potent, selective A3 adenosine receptor agonist with Ki of 0.33 nM, 2500- and 1400-fold selectivity over A1 and A2a receptors. |
| PC-63144 |
AZD-4635
|
1321514-06-0 |
AZD-4635 (HTL 1071) is a potent, selective and orally available adenosine 2A receptor (A2AR) inhibitor with Ki of 1.7 nM, > 30-fold selectivity over other adenosine receptors. |
| PC-70072 |
ST-1535
|
496955-42-1 |
ST1535 is a potent, selective A2A adenosine receptor antagonist with Ki of 6.6 nM. |
| PC-20111 |
ASP5854
|
851087-60-0 |
ASP5854 (ASP-5854) is a potent adenosine A(1) and A(2A) receptor dual antagonist with binding Ki of 9.03 and 1.76 nM for human A(1) and A(2A) receptors, respectively. |
| PC-20110 |
SCH-442416
|
316173-57-6 |
SCH-442416 (SCH442416) is a potent, selective and brain-penetrant antagonist of adenosine A2A receptor (A2AR) with Ki 0.048 nM and 0.5 nM for human and rat A2AR, respectively. |
