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TRR469

Chemical Structure : TRR469

CAS No.: 1394867-58-3

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TRR469 (TRR-469, TRR 469)

Catalog No.: PC-21513Not For Human Use, Lab Use Only.

TRR469 is a potent, selective adenosine A1 receptor (A1AR) positive allosteric modulator with pKb of 5.36, exhibits anti-nociceptive properties in acute and neuropathic pain models in mice.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    TRR469 is a potent, selective adenosine A1 receptor (A1AR) positive allosteric modulator with pKb of 5.36, exhibits anti-nociceptive properties in acute and neuropathic pain models in mice.

    Physicochemical Properties

    M.Wt 506.04
    Formula C28H25ClFN3OS
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (2-Amino-4-[(4-(phenyl)piperazin-1-yl)methyl]-5-(4-fluorophenyl)thiophen-3-yl)-(4-chlorophenyl)methanone

    References

    1. Vincenzi F, et al. Neuropharmacology. 2016 Dec;111:283-292.

    2. Romeo Romagnoli, et al. J Med Chem. 2012 Sep 13;55(17):7719-35.

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