| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-35841 |
AB928
|
2239273-34-6 |
Etrumadenant (AB928) is a potent, dual antagonist of the A2aR and A2bR adenosine receptors with Kb of 1.5 and 2.0 nM, respectively. |
| PC-35779 |
PBF509
|
1337962-47-6 |
PBF509 (Taminadenant, PBF-509, NIR 178) is a novel selective and potent Adenosine A2A Receptor (A2AR) antagonist, antagonizes A2AR agonist-mediated cAMP accumulation and impedance responses with KB values of 72.8 and 8.2 nM, respectively. |
| PC-43007 |
2-Cl-IB-MECA
|
163042-96-4 |
2-Cl-IB-MECA (Chloro-IB-MECA, CF-102, Namodenoson) is a potent, selective A3 adenosine receptor agonist with Ki of 0.33 nM, 2500- and 1400-fold selectivity over A1 and A2a receptors. |
| PC-63144 |
AZD-4635
|
1321514-06-0 |
AZD-4635 (HTL 1071) is a potent, selective and orally available adenosine 2A receptor (A2AR) inhibitor with Ki of 1.7 nM, > 30-fold selectivity over other adenosine receptors. |
| PC-38488 |
CGS-15943
|
104615-18-1 |
CGS-15943 is a potent, non-xanthine adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively. |
| PC-38365 |
Inupadenant
|
2246607-08-7 |
Inupadenant (EOS-850, EOS100850) is a non brain-penetrant, potent and highly selective small molecule antagonist of adenosine A2a receptor (A2AR), shows activity at the high adenosine concentrations found in tumors. |
| PC-38014 |
MIPS521
|
1146188-19-3 |
MIPS521 (MIPS-521) is a potent, positive allosteric modulator (PAM) of adenosine receptor (A1R). |
