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Cat. No. Product Name CAS No. Information
PC-35841

AB928

2239273-34-6 Etrumadenant (AB928) is a potent, dual antagonist of the A2aR and A2bR adenosine receptors with Kb of 1.5 and 2.0 nM, respectively.
PC-35779

PBF509

1337962-47-6 PBF509 (Taminadenant, PBF-509, NIR 178) is a novel selective and potent Adenosine A2A Receptor (A2AR) antagonist, antagonizes A2AR agonist-mediated cAMP accumulation and impedance responses with KB values of 72.8 and 8.2 nM, respectively.
PC-43007

2-Cl-IB-MECA

163042-96-4 2-Cl-IB-MECA (Chloro-IB-MECA, CF-102, Namodenoson) is a potent, selective A3 adenosine receptor agonist with Ki of 0.33 nM, 2500- and 1400-fold selectivity over A1 and A2a receptors.
PC-63144

AZD-4635

1321514-06-0 AZD-4635 (HTL 1071) is a potent, selective and orally available adenosine 2A receptor (A2AR) inhibitor with Ki of 1.7 nM, > 30-fold selectivity over other adenosine receptors.
PC-38488

CGS-15943

104615-18-1 CGS-15943 is a potent, non-xanthine adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.
PC-38365

Inupadenant

2246607-08-7 Inupadenant (EOS-850, EOS100850) is a non brain-penetrant, potent and highly selective small molecule antagonist of adenosine A2a receptor (A2AR), shows activity at the high adenosine concentrations found in tumors.
PC-38014

MIPS521

1146188-19-3 MIPS521 (MIPS-521) is a potent, positive allosteric modulator (PAM) of adenosine receptor (A1R).

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