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Request The Product List ofAdenosine Receptor Adenosine Receptor

Cat. No. Product Name Information
PC-42717

Vipadenant

A2AR antagonist

Vipadenant (BIIB014) is a potent and selective A2A adenosine receptor antagonist with Ki of 1.3 nM.
PC-42729

Preladenant

A2AR antagonist

Preladenant (SCH420814) is a potent and highly selective adenosine A2A receptor competitive antagonist with Ki of 1.1 nM.
PC-42728

Istradefylline

A2AR antagonist

Istradefylline (KW6002) is a potent and highly selective A2A receptor antagonist with Ki of 2.2 nM.
PC-45527

APNEA

A3AR agonist

APNEA is a non-selective agonist of adenosine A3 receptor, has a high affinity for the adenosine A1 and A3 receptors.
PC-45624

AB-MECA

A3AR agonist

AB-MECA is a high affinity A3 adenosine receptor (A3AR) agonist with binding Ki of 430.5 nM for human A3 receptors in CHO cells.
PC-23655

Regadenoson

A2A receptor antagonist

Regadenoson (CVT-3146) is a potent, selective A2A adenosine receptor agonist, and short-acting coronary vasodilator.
PC-23389

SLV320

Adenosine A1 receptor antagonist

Derenofylline (SLV320) is a potent, selective and orally active adenosine A1 receptor antagonist with Ki values of 1 nM, 200 nM and 398 nM for human A1, A3 and A2A receptors respectively.
PC-23365

TC-G 1004

A2A receptor antagonist

TC-G 1004 is a potent, selective orally active A2A adenosine receptor (A2A R) antagonist, with Ki values of 0.44 nM and 80 nM for hA2A and hA1, respectively.
PC-22840

DPCPX

Adenosine A1 receptor antagonist

DPCPX (PD116948) is a highly potent and selective adenosine A1 receptor antagonist with Ki of 0.46 nM, >500-fold selective over A2 receptor.
PC-22838

AR-001

Adenosine A1 receptor agonist

AR-001 is a selective adenosine A1 receptor agonist with EC50 of 9.35 uM in HEK293-aeqα15/ADORA1 cells, increases adenosine A1 receptor expression and mRNA level in the hypothalamus of mice, exhibits hypnotic efficacy.
PC-22753

MRS-1706

A2BR antagonist

MRS-1706 (MRS1706) is a potent and selective adenosine A2B receptor (A2BR) inverse agonist / antagonist with Ki of 1.39 nM, >100-fold selective over A2A, A1 and A3 receptors.
PC-22524

MRS1754

A2BR antagonist

MRS 1754 is a potent, adenosine receptor A2BAR selective antagonist with Ki of 1.97 nM, 205-, 255-, and 289-fold selective for the human A2BARs vs. human A1/A2A/A3 ARs, respectively.

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