| Cat. No. |
Product Name |
Information |
| PC-44125 |
Capadenoson
A1AR agonist
|
Capadenoson (BAY68-4986) is a selective agonist of adenosine-A1 receptor (A1AR). |
| PC-42771 |
Tozadenant
A2AR antagonist
|
Tozadenant (SYN115) is a potent, selective adenosine 2A receptor (A2AR) antagonist with Ki of 11.5 nM. |
| PC-45585 |
GR-79236
A1AR agonist
|
GR-79236 is a potent and selective Adenosine A1 receptor agonist with Ki of 3.1 nM. |
| PC-42717 |
Vipadenant
A2AR antagonist
|
Vipadenant (BIIB014) is a potent and selective A2A adenosine receptor antagonist with Ki of 1.3 nM. |
| PC-42729 |
Preladenant
A2AR antagonist
|
Preladenant (SCH-420814, MK-3814) is a potent and highly selective adenosine A2A receptor competitive antagonist with Ki of 1.1 nM. |
| PC-42728 |
Istradefylline
A2AR antagonist
|
Istradefylline (KW-6002) is a potent and highly selective A2A receptor antagonist with Ki of 2.2 nM. |
| PC-45527 |
APNEA
A3AR agonist
|
APNEA is a non-selective agonist of adenosine A3 receptor, has a high affinity for the adenosine A1 and A3 receptors. |
| PC-45624 |
AB-MECA
A3AR agonist
|
AB-MECA is a high affinity A3 adenosine receptor (A3AR) agonist with binding Ki of 430.5 nM for human A3 receptors in CHO cells. |
| PC-25476 |
MIPS2719
A1AR antagonist
|
MIPS2719 is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR)with pKB value of 8.2, selective for the A1AR over the A2AAR. |
| PC-25475 |
MIPS2712
A1AR antagonist
|
MIPS2712 is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR)with pKB value of 8.0, >100-fold selective for the A1AR over the A2AAR. |
| PC-25474 |
NECA
Adenosine receptor agonist
|
NECA (5'-N-Ethylcarboxamidoadenosine) is a nonselective adenosine receptor agonist. |
| PC-25473 |
DU172
A1AR antagonist
|
DU172 (Compound 23b) is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR), inhibits [3H]DPCPX binding to A1AR with IC50 of 21 nM, 132-fold more selective for the A1AR over the A2AAR. |
