| Cat. No. |
Product Name |
Information |
| PC-45527 |
APNEA
A3AR agonist
|
APNEA is a non-selective agonist of adenosine A3 receptor, has a high affinity for the adenosine A1 and A3 receptors. |
| PC-45624 |
AB-MECA
A3AR agonist
|
AB-MECA is a high affinity A3 adenosine receptor (A3AR) agonist with binding Ki of 430.5 nM for human A3 receptors in CHO cells. |
| PC-22524 |
MRS1754
A2BR antagonist
|
MRS 1754 is a potent, adenosine receptor A2BAR selective antagonist with Ki of 1.97 nM, 205-, 255-, and 289-fold selective for the human A2BARs vs. human A1/A2A/A3 ARs, respectively. |
| PC-22361 |
LUF5834
A2AR agonist
|
LUF5834 is a potent, selective, non-adenosine adenosine A1 receptor adenosine receptor (A2BR) partial agonist with EC50 of 12 nM (hA2B), 45-fold selective over hA3, also shows high affinity with Ki of 2.6 nM and 28 nM for hA1 and hA2A, respectively. |
| PC-22194 |
CF102
A3AR agonist
|
Namodenoson (2-Cl-IB-MECA, CF-102) is a potent, selective A3 adenosine receptor (A3AR) agonist with Ki of 0.33 nM, displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively. |
| PC-22193 |
CF101
A3AR agonist
|
Piclidenoson (IB-MECA, CF101) is a first-in-class, orally active and selective A3 adenosine receptor (A3AR) agonist, shows antiproliferative effect and induces apoptosis in multiple cancer cell types like melanoma, leukemia. |
| PC-22012 |
CVT-7124
A2B adenosine receptor inhibitor
|
CVT-7124 (CVT7124) is a highly potent, selective A2B adenosine receptor antagonist with Ki of 6 nM (hA2B), >830-fold selective over A1, A2A and A3 receptors. |
| PC-21511 |
MRS7469
A1AR agonist
|
MRS7469 is a potent and selective orthosteric A1 adenosine receptor (A1AR) agonist with Ki of 2.14 nM, >2000-fold selective for A1AR over other adenosine receptors. |
| PC-20644 |
VUF-5574
A3 adenosine antagonist
|
VUF-5574 (VUF5574) is a potent, selective A3 adenosine receptor antagonist with high affinity (Ki=4.03 nM, human A3 receptor). |
| PC-20643 |
OT-7999
A3 adenosine antagonist
|
OT-7999 (OT7999) is a potent and selective adenosine A3 receptor antagonist with Ki of 0.61 nM (human A3 receptor) in radioligand binding assays. |
| PC-20641 |
MRS1191
A3 adenosine antagonist
|
MRS1191 (MRS-1191) is a potent and selective A3 adenosine receptor antagonist with Ki of 32 nM, shows no acitivity against A2A, A2B, A1 receptors (Ki>10 uM). |
| PC-20110 |
SCH-442416
A2AR antagonist
|
SCH-442416 (SCH442416) is a potent, selective and brain-penetrant antagonist of adenosine A2A receptor (A2AR) with Ki 0.048 nM and 0.5 nM for human and rat A2AR, respectively. |
