Cat. No. |
Product Name |
Information |
PC-20111 |
ASP5854
A1R/A2R dual inhibitor
|
ASP5854 (ASP-5854) is a potent adenosine A(1) and A(2A) receptor dual antagonist with binding Ki of 9.03 and 1.76 nM for human A(1) and A(2A) receptors, respectively. |
PC-20110 |
SCH-442416
A2AR antagonist
|
SCH-442416 (SCH442416) is a potent, selective and brain-penetrant antagonist of adenosine A2A receptor (A2AR) with Ki 0.048 nM and 0.5 nM for human and rat A2AR, respectively. |
PC-20101 |
GS 6201
A2B adenosine receptor inhibitor
|
GS-6201 (CVT-6883, GS6201) is a specific and selective A2B adenosine receptor antagonist with Ki of 22 nM, >50-fold selectivity over A3, A1 and A2A receptors. |
PC-20100 |
JNJ-40255293
Adenosine A2A/A1 inhibitor
|
JNJ-40255293 (JNJ 40255293) is a potent, dual adenosine A2A/A1 receptor antagonist with Ki of 6.8/42 nM, respectively. |
PC-49545 |
PSB-603
A(2b)R antagonist
|
PSB-603 is a potent, selective adenosine A2B receptor antagonist with Ki of 0.553 nM, >17000-fold selectivity over other adenosine receptors (A1, A2A and A3 receptors). |
PC-49354 |
M1069
A2A A2B antagonist
|
M1069 (M-1069) is a potent, dual antagonist of the A2A and A2B adenosine receptors, with selectivity of >100 fold against the A1 and A3 receptors. |
PC-38488 |
CGS-15943
Adenosine receptor inhibitor
|
CGS-15943 is a potent, non-xanthine adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively. |
PC-38365 |
Inupadenant
A2AR antagonist
|
Inupadenant (EOS-850, EOS100850) is a non brain-penetrant, potent and highly selective small molecule antagonist of adenosine A2a receptor (A2AR), shows activity at the high adenosine concentrations found in tumors. |
PC-36102 |
Taminadenant
|
Taminadenant is an adenosine receptor A2a antagonist.. |
PC-36101 |
KH-176
|
KH-176 (KH176, Sonlicromanol) is a smal molecule ROS-redox modulator, effectively reduces increased cellular ROS levels and protects OXPHOS deficient primary cells against redox perturbation by targeting the Thioredoxin/Peroxiredoxin system. |
PC-35973 |
MRS1186
|
MRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM.. |
PC-35507 |
MSX-3 hydrate
|
MSX-3 hydrate is a potent, specific adenosine A2A receptor (A2AR) antagonist.. |