You are here:Home-Chemical Inhibitors & Agonists-GPCR-Adenosine Receptor

Request The Product List ofAdenosine Receptor Adenosine Receptor

Cat. No. Product Name Information
PC-20111

ASP5854

A1R/A2R dual inhibitor

ASP5854 (ASP-5854) is a potent adenosine A(1) and A(2A) receptor dual antagonist with binding Ki of 9.03 and 1.76 nM for human A(1) and A(2A) receptors, respectively.
PC-20110

SCH-442416

A2AR antagonist

SCH-442416 (SCH442416) is a potent, selective and brain-penetrant antagonist of adenosine A2A receptor (A2AR) with Ki 0.048 nM and 0.5 nM for human and rat A2AR, respectively.
PC-20101

GS 6201

A2B adenosine receptor inhibitor

GS-6201 (CVT-6883, GS6201) is a specific and selective A2B adenosine receptor antagonist with Ki of 22 nM, >50-fold selectivity over A3, A1 and A2A receptors.
PC-20100

JNJ-40255293

Adenosine A2A/A1 inhibitor

JNJ-40255293 (JNJ 40255293) is a potent, dual adenosine A2A/A1 receptor antagonist with Ki of 6.8/42 nM, respectively.
PC-49545

PSB-603

A(2b)R antagonist

PSB-603 is a potent, selective adenosine A2B receptor antagonist with Ki of 0.553 nM, >17000-fold selectivity over other adenosine receptors (A1, A2A and A3 receptors).
PC-49354

M1069

A2A A2B antagonist

M1069 (M-1069) is a potent, dual antagonist of the A2A and A2B adenosine receptors, with selectivity of >100 fold against the A1 and A3 receptors.
PC-38488

CGS-15943

Adenosine receptor inhibitor

CGS-15943 is a potent, non-xanthine adenosine receptor antagonist with Ki values of 3.5, 4.2, 16 and 51 nM for human A1, A2A, A2B and A3 receptors respectively.
PC-38365

Inupadenant

A2AR antagonist

Inupadenant (EOS-850, EOS100850) is a non brain-penetrant, potent and highly selective small molecule antagonist of adenosine A2a receptor (A2AR), shows activity at the high adenosine concentrations found in tumors.
PC-36102

Taminadenant

Taminadenant is an adenosine receptor A2a antagonist..
PC-36101

KH-176

KH-176 (KH176, Sonlicromanol) is a smal molecule ROS-redox modulator, effectively reduces increased cellular ROS levels and protects OXPHOS deficient primary cells against redox perturbation by targeting the Thioredoxin/Peroxiredoxin system.
PC-35973

MRS1186

MRS1186 (MRS-1186) is a potent and selective human Adenosine A3 receptor (hA3AR) antagonist with Ki of 7.66 nM..
PC-35507

MSX-3 hydrate

MSX-3 hydrate is a potent, specific adenosine A2A receptor (A2AR) antagonist..

Request The Product List

* Indicates a Required FieldYour information is safe with us.

  • *Product List:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Country:
  • Additional Information:

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com