| Cat. No. |
Product Name |
Information |
| PC-25472 |
FSCPX
A1AR antagonist
|
FSCPX is a potent, selective and irreversible antagonist of A1-adenosine receptor (A1AR), FSCPX (5 uM) completely reverses the increase in K+ current of guinea pig atrial myocytes. |
| PC-25471 |
LUF7602
A3AR antagonist
|
LUF7602 is a selective, covalent antagonist of A3 adenosine receptor (A3AR) with pKi of 7.5. |
| PC-25169 |
VG081821AC
A2A receptor antagonist
|
VG081821AC (VG081821 acetate) is a potent, selective, orally active A2A adenosine receptor antagonist with binding Ki of 0.85 nM, >300-fold selective over A1, A2B, and A3 receptors. |
| PC-25168 |
VG081821
A2A receptor antagonist
|
VG081821 is a potent, selective, orally active A2A adenosine receptor antagonist with binding Ki of 0.85 nM, >300-fold selective over A1, A2B, and A3 receptors. |
| PC-24974 |
A1R PAM 56
A1R PAM
|
A1R PAM 56 is a potent, selective positive allosteric modulator of A1 adenosine receptor (A1R), modulates NECA affinity (pK) and potency (pEC50). |
| PC-24373 |
VCP746
A1AR agonist
|
VCP746 is a selective, hybrid molecule A1 adenosine receptor (A1AR) biased agonist with Ki of 60 nM, and pEC50 of 9.05 in FlpIn-CHO cells stably expressing the A1AR. |
| PC-24291 |
HZ-086
A2AR inhibitor
|
HZ-086 is a potent and selective inhibitor of adenosine A2A receptor (A2AR) with Ki of 1.4 nM (hA2A), >250-fold selective over A1R and A3R. |
| PC-24196 |
Zaladenant
A2a receptor inhibitor
|
Zaladenant is a potent, selective adenosine A2a receptor inhibitor with IC50 of 0.23 nM. |
| PC-23909 |
FM101
A3AR inhibitor
|
FM101 is a highly potent and selective antagonist of A3 adenosine receptor (A3AR), selectively binds to human A3AR with Ki of 1.44 nM. |
| PC-23655 |
Regadenoson
A2A receptor antagonist
|
Regadenoson (CVT-3146) is a potent, selective A2A adenosine receptor agonist, and short-acting coronary vasodilator. |
| PC-23365 |
TC-G 1004
A2A receptor antagonist
|
TC-G 1004 is a potent, selective orally active A2A adenosine receptor (A2A R) antagonist, with Ki values of 0.44 nM and 80 nM for hA2A and hA1, respectively. |
| PC-22838 |
AR-001
Adenosine A1 receptor agonist
|
AR-001 is a selective adenosine A1 receptor agonist with EC50 of 9.35 uM in HEK293-aeqα15/ADORA1 cells, increases adenosine A1 receptor expression and mRNA level in the hypothalamus of mice, exhibits hypnotic efficacy. |
