| Cat. No. |
Product Name |
Information |
| PC-45527 |
APNEA
A3AR agonist
|
APNEA is a non-selective agonist of adenosine A3 receptor, has a high affinity for the adenosine A1 and A3 receptors. |
| PC-45624 |
AB-MECA
A3AR agonist
|
AB-MECA is a high affinity A3 adenosine receptor (A3AR) agonist with binding Ki of 430.5 nM for human A3 receptors in CHO cells. |
| PC-28314 |
IHCH-3064
A2AR/HDAC inhibitor
|
IHCH-3064 is a potent, dual-targeting adenosine A2A receptor (A2AR) antagonist and HDAC inhibitor with Ki of 2.2 nM (A2AR) and IC50 of 80.2 nM (HDAC1) respectively. |
| PC-28312 |
IHCH-3185
A2AR/HDAC inhibitor
|
IHCH-3185 is a potent, dual-targeting adenosine A2A receptor (A2AR) antagonist and HDAC inhibitor with Ki of 7.6 nM (A2AR) and IC50 of 102.9 nM (HDAC1) respectively. |
| PC-27870 |
N6-cyclopentyladenosine
Adenosine A1 receptor agonist
|
N6-Cyclopentyladenosine (CPA) is a high affinity, selective adenosine A1 receptor (A1R) agonist with Ki of 2.3 nM, 790 nM and 43 nM for human A1, A2A and A3 receptors, respectively. |
| PC-26915 |
INCB106385
Adenosine A2A/A2B receptor antagonist
|
INCB106385 is a potent, selective dual A2A/A2B adenosine receptor antagonist. |
| PC-26045 |
A2AR antagonist P625
A2AR antagonist
|
A2AR antagonist P625 is a highly potent, selective adenosine A2A receptor (A2AR) antagonist with Ki of 15.1 nM (human cloned A2AR), ameliorates EAE symptoms by attenuating neuroinflammation and demyelination. |
| PC-26044 |
A2AR antagonist P400
A2AR antagonist
|
A2AR antagonist P400 is a highly potent, selective adenosine A2A receptor (A2AR) antagonist with Ki of 5.3 fM (human cloned A2AR), ameliorates EAE symptoms by attenuating neuroinflammation and demyelination. |
| PC-26034 |
IDPU
A2AR antagonist
|
IDPU is a high potent, selective Adenosine A2A receptor (A2AR) antagonist with Ki of 0.0038 nM, has 737-fold selectivity over A1R. |
| PC-25685 |
LJ-4378
A2AAR agonist, A3AR antagonist
|
LJ-4378 is a dual-acting ligand with A2AAR agonist (EC50=80.3 nM for cAMP formation, binding Ki=7.19 nM) and A3 adenosine receptor (A3AR, binding Ki=11.8 nM) antagonist activity. |
| PC-25476 |
MIPS2719
A1AR antagonist
|
MIPS2719 is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR)with pKB value of 8.2, selective for the A1AR over the A2AAR. |
| PC-25475 |
MIPS2712
A1AR antagonist
|
MIPS2712 is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR)with pKB value of 8.0, >100-fold selective for the A1AR over the A2AAR. |
