| Cat. No. |
Product Name |
Information |
| PC-26034 |
IDPU
A2AR antagonist
|
IDPU is a high potent, selective Adenosine A2A receptor (A2AR) antagonist with Ki of 0.0038 nM, has 737-fold selectivity over A1R. |
| PC-25759 |
P626
A2AR/A2BR antagonist
|
P626 is a potent, selective dual adenosine A2A/A2B receptor (A2AR/A2BR) antagonist with IC50 of 5.73 nM and 34 nM at both hA2AAR and hA2BAR (cAMP assay), with no significant acitivity against hA1AR and hA3AR. |
| PC-25685 |
LJ-4378
A2AAR agonist, A3AR antagonist
|
LJ-4378 is a dual-acting ligand with A2AAR agonist (EC50=80.3 nM for cAMP formation, binding Ki=7.19 nM) and A3 adenosine receptor (A3AR, binding Ki=11.8 nM) antagonist activity. |
| PC-25476 |
MIPS2719
A1AR antagonist
|
MIPS2719 is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR)with pKB value of 8.2, selective for the A1AR over the A2AAR. |
| PC-25475 |
MIPS2712
A1AR antagonist
|
MIPS2712 is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR)with pKB value of 8.0, >100-fold selective for the A1AR over the A2AAR. |
| PC-25474 |
NECA
Adenosine receptor agonist
|
NECA (5'-N-Ethylcarboxamidoadenosine) is a nonselective adenosine receptor agonist. |
| PC-25473 |
DU172
A1AR antagonist
|
DU172 (Compound 23b) is a potent, selective, covalent, irreversible antagonist of A1 adenosine receptor (A1AR), inhibits [3H]DPCPX binding to A1AR with IC50 of 21 nM, 132-fold more selective for the A1AR over the A2AAR. |
| PC-25472 |
FSCPX
A1AR antagonist
|
FSCPX is a potent, selective and irreversible antagonist of A1-adenosine receptor (A1AR), FSCPX (5 uM) completely reverses the increase in K+ current of guinea pig atrial myocytes. |
| PC-25471 |
LUF7602
A3AR antagonist
|
LUF7602 is a selective, covalent antagonist of A3 adenosine receptor (A3AR) with pKi of 7.5. |
| PC-25169 |
VG081821AC
A2A receptor antagonist
|
VG081821AC (VG081821 acetate) is a potent, selective, orally active A2A adenosine receptor antagonist with binding Ki of 0.85 nM, >300-fold selective over A1, A2B, and A3 receptors. |
| PC-25168 |
VG081821
A2A receptor antagonist
|
VG081821 is a potent, selective, orally active A2A adenosine receptor antagonist with binding Ki of 0.85 nM, >300-fold selective over A1, A2B, and A3 receptors. |
| PC-24974 |
A1R PAM 56
A1R PAM
|
A1R PAM 56 is a potent, selective positive allosteric modulator of A1 adenosine receptor (A1R), modulates NECA affinity (pK) and potency (pEC50). |
