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Chemical Structure : LUF5834
Catalog No.: PC-22361Not For Human Use, Lab Use Only.
LUF5834 is a potent, selective, non-adenosine adenosine A1 receptor adenosine receptor (A2BR) partial agonist with EC50 of 12 nM (hA2B), 45-fold selective over hA3, also shows high affinity with Ki of 2.6 nM and 28 nM for hA1 and hA2A, respectively.
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LUF5834 is a potent, selective, non-adenosine adenosine A1 receptor adenosine receptor (A2BR) partial agonist with EC50 of 12 nM (hA2B), 45-fold selective over hA3.
LUF5834 also shows high affinity with Ki of 2.6 nM and 28 nM for hA1 and hA2A, respectively.
| M.Wt | 348.38 | |
| Formula | C17H12N6OS | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Beukers MW, et al. J Med Chem. 2004 Jul 15;47(15):3707-9.
2. Urmaliya VB, et al. J Cardiovasc Pharmacol. 2009 May;53(5):424-33.
3. Lane JR, et al. Biochem Pharmacol. 2010 Oct 15;80(8):1180-9.
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