| Cat. No. |
Product Name |
CAS No. |
Information |
| PC-49624 |
SGC-CAMKK2-1N
|
|
SGC-CAMKK2-1N is the negative control compound of the CaMKK2 inhibitor SGC-CAMKK2-1 (Catalog# PC-49623), shows significantly less potent with CAMKK2 (IC50=27 uM). |
| PC-49623 |
SGC-CAMKK2-1
|
2561494-76-4 |
SGC-CAMKK2-1 is a potent, selective chemical probe inhibitor that targets CAMKK2 with enzyme IC50 of 30 nM. |
| PC-49436 |
NCS-382
|
520505-01-5 |
NCS-382 is a a gamma-hydroxybutyrate receptor (GHBR) antagonist, brain-penetrating high nanomolar-affinity ligand selective for the CaMKIIα hub domain, possesses antagonistic properties |
| PC-49435 |
Ph-HTBA
|
2368927-41-5 |
Ph-HTBA is a mid-nanomolar affinity (Ki=78nM), brain permeable ligand of CaMKIIα hub domain binding site. |
| PC-72972 |
AS105
|
1026029-18-4 |
AS105 (AS-105) is a highly potent, ATP-competitive CaMKII inhibitor, inhibits CaMKIIδ with IC50 of 8 nM, Ki of 3 nM. |
| PC-72971 |
GS-680
|
|
GS-680 (GS680) is a novel selective and ATP-competitive CaMKII inhibitor with biochemical IC50 of 2.3 and 15.9 nM against CaMKIIδ and CaMKIIα, respectively. |
| PC-72970 |
RA608
|
|
RA608 (RA-608) is a potent, selective, ATP-competitive, orally available CaMKII inhibitor, inhibits human CaMKIIδ, CaMKIIɣ, CaMKIIα, and CaMKIIβ with IC50 of 22, 51, 121, and 1135 nM, respectively. |
