Cat. No. |
Product Name |
Information |
PC-43468 |
KN-62
CaMK II inhibitor
|
KN-62 is a specific inhibitor of Ca2+/calmodulin-dependent protein kinase II (CaMK II) with Ki of 900 nM for rat brain CaMK II. |
PC-63352 |
CAMKK2 inhibitor 4t
CAMKK2 inhibitor
|
CAMKK2 inhibitor 4t is a potent, selective, orally available, brain-penetrant CAMKK2 inhibitor with pIC50 of 8.5. |
PC-45723 |
STO-609
CaMKK inhibitor
|
STO-609 is a selective and cell-permeable inhibitor of CaM-KK, inhibits recombinant CaM-KKα and CaM-KKβ with Ki of 80 and 15 ng/ml. |
PC-45443 |
CaMKII-IN-1
CaMKII inhibitor
|
CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM. |
PC-23447 |
TRIB2 inhibitor 1 hydrochloride
TRIB2 inhibitor
|
TRIB2 inhibitor 1 hydrochloride is a small-molecule binder and inhibitor of Tribbles pseudokinase 2 (TRIB2), downregulates TRIB2 levels at micromolar concentration. |
PC-23446 |
TRIB2 inhibitor 1
TRIB2 inhibitor
|
TRIB2 inhibitor 1 is a small-molecule binder and inhibitor of Tribbles pseudokinase 2 (TRIB2), downregulates TRIB2 levels at micromolar concentration. |
PC-23411 |
DXL-A-24
CaMKIIα inhibitor
|
DXL-A-24 is a spirocyclopiperazinium salt compound with antinociceptive effect, alleviates neuropathic pain by inhibiting CGRP expression, inhibits CaMKIIα phosphorylation. |
PC-21505 |
SMP-114
CaMKII inhibitor
|
SMP-114 (Rimacalib) is a potent, specific and orally available CaMKII inhibitor with potential for treatment of rheumatoid arthritis. |