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Chemical Structure : CaMKII-IN-1
CAS No.: 1208123-85-6
Catalog No.: PC-45443Not For Human Use, Lab Use Only.
CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $138 | In stock | |
| 10 mg | $228 | In stock | |
| 25 mg | $398 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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CaMKII-IN-1 is a potent and highly selective CaMKII inhibitor with IC50 of 63 nM.
CaMKII-IN-1 shows no inhibitory effect for CaMKIV, MLCK, p38α, Akt1, PKC etc.
CaMKII-IN-1 shows 25-fold higher potency than KN-93.
| M.Wt | 548.0988 | |
| Formula | C29H30ClN5O2S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 54 mg/mL |
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| Chemical Name/SMILES |
Benzenesulfonamide, 3-chloro-2-methyl-N-[5,6,7,8-tetrahydro-2-[(2-phenylethyl)amino]-6-(phenylmethyl)pyrido[4,3-d]pyrimidin-4-yl]- |
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1. Asano S, et al. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6696-8.
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