CVT-7124 | A2B adenosine receptor inhibitor

Chemical Structure : CVT-7124

CVT-7124 (CVT7124)

Catalog No.: PC-22012Not For Human Use, Lab Use Only.

CVT-7124 (CVT7124) is a highly potent, selective A2B adenosine receptor antagonist with Ki of 6 nM (hA2B), >830-fold selective over A1, A2A and A3 receptors.

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Biological Activity

CVT-7124 (CVT7124) is a highly potent, selective A2B adenosine receptor antagonist with Ki of 6 nM (hA2B), >830-fold selective over A1, A2A and A3 receptors.
CVT-7124 blocks the release of interleukin-6 and monocyte chemotactic protein-1 from bronchial smooth muscle cells (BSMC).

Physicochemical Properties

M.Wt	404.35
Formula	C18H15F3N6O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	1-ethyl-8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazol-4-yl)-3,7-dihydro-1H-purine-2,6-dione

References

1. Rao V Kalla, et al. Bioorg Med Chem Lett. 2008 Feb 15;18(4):1397-401.

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CVT-7124 (CVT7124)

Biological Activity

Physicochemical Properties

References

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