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TC-G 1004

Chemical Structure : TC-G 1004

CAS No.: 1061747-72-5

TC-G 1004 (TC-G1004)

Catalog No.: PC-23365Not For Human Use, Lab Use Only.

TC-G 1004 is a potent, selective orally active A2A adenosine receptor (A2A R) antagonist, with Ki values of 0.44 nM and 80 nM for hA2A and hA1, respectively.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

TC-G 1004 is a potent, selective orally active A2A adenosine receptor (A2A R) antagonist, with Ki values of 0.44 nM and 80 nM for hA2A and hA1, respectively.

Physicochemical Properties

M.Wt 421.51
Formula C22H27N7O2
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

N-(2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(6-(4-methoxypiperidin-1-yl)pyridin-2-yl)pyrimidin-4-yl)acetamide

References

1. Xiaohu Zhang, et al. 2008 Nov 27;51(22):7099-110.

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