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Chemical Structure : MRS1754
CAS No.: 264622-58-4
Catalog No.: PC-22524Not For Human Use, Lab Use Only.
MRS 1754 is a potent, adenosine receptor A2BAR selective antagonist with Ki of 1.97 nM, 205-, 255-, and 289-fold selective for the human A2BARs vs. human A1/A2A/A3 ARs, respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $98 | In stock | |
| 10 mg | $158 | In stock | |
| 25 mg | $278 | In stock | |
| 50 mg | $478 | In stock | |
| 100 mg | Get quote |
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MRS 1754 is a potent, adenosine receptor A2BAR selective antagonist with Ki of 1.97 nM, 205-, 255-, and 289-fold selective for the human A2BARs vs. human A1/A2A/A3 ARs, respectively.
| M.Wt | 486.53 | |
| Formula | C26H26N6O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
8-[4-[((4-cyanophenyl)carbamoylmethyl)oxy]phenyl]-1,3-di(n-propyl) xanthine |
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1. Zizzo MG, et al. Br J Pharmacol. 2006 Aug;148(7):956-63.
2. Jacobson KA. Drug Dev Res. 2001 Jan-Feb;52(1-2):178-186.
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