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Chemical Structure : MRS7935
Catalog No.: PC-21510Not For Human Use, Lab Use Only.
MRS7935 is a potent, selective positive allosteric modulator (PAM) of A1 adenosine receptor (A1AR) with EC50 of 1.43 uM.
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MRS7935 is a potent, selective positive allosteric modulator (PAM) of A1 adenosine receptor (A1AR) with EC50 of 1.43 uM.
MRS7935 displays no functional activity at hA2A, hA2B, and hA3ARs at 30 μM.
MRS7935 (1 uM) enhances the functional activity of A1AR agonist Cl-ENBA.
MRS7935 does not enhance hypothermia in vivo induced by either adenosine or a selective A1AR agonist.
| M.Wt | 443.94 | |
| Formula | C24H20ClF2NOS | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Paola Oliva, et al. ACS Medicinal Chemistry Letters, 2023.
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