CGRP Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-27352	PRT-064040 CGRP antagonist	PRT-064040 is a potent, selective calcitonin gene-related peptide receptor (CGRP) antagonist with binding Ki of 26.67 pM (human CGRP receptor), effectively inhibits human αCGRP-induced cAMP production with IC50 of 22.29 pM.
PC-24985	CGRP receptor antagonist 15 CGRP inhibitor	CGRP receptor antagonist 15 is a highly potent, orally bioavailable calcitonin gene-related peptide (CGRP) receptor antagonist with Ki of 0.029 nM and cAMP IC50 of 0.17 nM.
PC-24984	HTL22562 CGRP inhibitor	HTL22562 is a highly potent, selective, metabolically stable antagonist of calcitonin gene-related peptide (CGRP) receptor with pKi of 10.5 (human CGRP).
PC-21156	BMS-694153 CGRP antagonist	BMS-694153 is a potent, selective calcitonin gene-related peptide (CGRP) receptor antagonist with Ki of 0.013 nM for hCGRP (inhibition of 125I-CGRP binding in SK-N-MC cell membranes).

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