CGRP Receptor (inhibitors, antagonists, agonists)-ProbeChem.com

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Cat. No.	Product Name	Information
PC-24985	CGRP receptor antagonist 15 CGRP inhibitor	CGRP receptor antagonist 15 is a highly potent, orally bioavailable calcitonin gene-related peptide (CGRP) receptor antagonist with Ki of 0.029 nM and cAMP IC50 of 0.17 nM.
PC-24984	HTL22562 CGRP inhibitor	HTL22562 is a highly potent, selective, metabolically stable antagonist of calcitonin gene-related peptide (CGRP) receptor with pKi of 10.5 (human CGRP).
PC-24755	Cagrilintide acetate AMYR/CTR agonist	Cagrilintide acetate (AM833) is a long-acting amylin analogue as a nonselective amylin receptor (AMYR) and calcitonin G protein-coupled receptor (CTR) agonist with binding IC50 of 170 and 223 pM, and cAMP EC50 of 348 and 287 pM for hAMY3R and hCTR respectively.
PC-24754	Cagrilintide AMYR/CTR agonist	Cagrilintide (AM833) is a long-acting amylin analogue as a nonselective amylin receptor (AMYR) and calcitonin G protein-coupled receptor (CTR) agonist with binding IC50 of 170 and 223 pM, and cAMP EC50 of 348 and 287 pM for hAMY3R and hCTR respectively.
PC-21156	BMS-694153 CGRP antagonist	BMS-694153 is a potent, selective calcitonin gene-related peptide (CGRP) receptor antagonist with Ki of 0.013 nM for hCGRP (inhibition of 125I-CGRP binding in SK-N-MC cell membranes).

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