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PRT-064040

Chemical Structure : PRT-064040

CAS No.:

PRT-064040 (PRT064040)

Catalog No.: PC-27352Not For Human Use, Lab Use Only.

PRT-064040 is a potent, selective calcitonin gene-related peptide receptor (CGRP) antagonist with binding Ki of 26.67 pM (human CGRP receptor), effectively inhibits human αCGRP-induced cAMP production with IC50 of 22.29 pM.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

PRT-064040 is a potent, selective calcitonin gene-related peptide receptor (CGRP) antagonist with binding Ki of 26.67 pM (human CGRP receptor), effectively inhibits human αCGRP-induced cAMP production with IC50 of 22.29 pM.

Physicochemical Properties

M.Wt
Formula
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

References

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