CGRP receptor antagonist 15

Chemical Structure : CGRP receptor antagonist 15

Catalog No.: PC-24985Not For Human Use, Lab Use Only.

CGRP receptor antagonist 15 is a highly potent, orally bioavailable calcitonin gene-related peptide (CGRP) receptor antagonist with Ki of 0.029 nM and cAMP IC50 of 0.17 nM.

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Biological Activity

CGRP receptor antagonist 15 is a highly potent, orally bioavailable calcitonin gene-related peptide (CGRP) receptor antagonist with Ki of 0.029 nM and cAMP IC50 of 0.17 nM.

Physicochemical Properties

M.Wt	529.62
Formula	C30H32FN5O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(2-((2R,5S)-2-(2-Cyanopropan-2-yl)-5-(3-fluorophenyl)pyrrolidin-1-yl)-2-oxoethyl)-3-methyl-4-((6-methyl-3-oxo-2,3-dihydropyridazin-4-yl)methyl)benzamide

References

1. Morita N, et al. J Med Chem. 2025 Jul 3. doi: 10.1021/acs.jmedchem.5c01127.

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