CCG 258001 |CAS:2055990-96-8 Probechem Biochemicals

Chemical Structure : CCG 258001

CCG 258001 (CCG258001;CCG-258001)

Catalog No.: PC-60588Not For Human Use, Lab Use Only.

CCG 258001 is a potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM.

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Biological Activity

CCG 258001 is a potent, relatively selective G protein-coupled receptor kinase GRK2 inhibitor with IC50 of 280 nM.
CCG 258001 displays >100-fold selectivity over GRK5, GRK1, PKA and ROCK1.

Physicochemical Properties

M.Wt	339.414
Formula	C20H22FN3O
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	5-(((3S,4R)-4-(4-fluorophenyl)-1-methylpiperidin-3-yl)methoxy)-1H-indazole

References

1. Bouley R, et al. Mol Pharmacol. 2017 Dec;92(6):707-717.

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CCG 258001 (CCG258001;CCG-258001)

Biological Activity

Physicochemical Properties

References

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