Chemical Structure : Takeda103A
CAS No.: 865609-72-9
Catalog No.: PC-38542Not For Human Use, Lab Use Only.
Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5.
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Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5.
M.Wt | 463.49 | |
Formula | C24H23F2N7O | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
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Chemical Name/SMILES |
N-[(2,6-Difluorophenyl)methyl]-3-[[[4-propyl-5-(4-pyrimidinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-benzamide |
1. Helen V Waldschmidt, et al. J Med Chem. 2016 Apr 28;59(8):3793-807.
2. Thal DM, et al. Mol Pharmacol. 2011;80:294–303.
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