Takeda103A | GRK2 inhibitor | Probechem Biochemicals

Chemical Structure : Takeda103A

CAS No.: 865609-72-9

Catalog No.: PC-38542Not For Human Use, Lab Use Only.

Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5.

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10 mg	$398	In stock
25 mg	$598	In stock
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Biological Activity

Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5.

M.Wt	463.49
Formula	C24H23F2N7O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-[(2,6-Difluorophenyl)methyl]-3-[[[4-propyl-5-(4-pyrimidinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-benzamide

1. Helen V Waldschmidt, et al. J Med Chem. 2016 Apr 28;59(8):3793-807.

2. Thal DM, et al. Mol Pharmacol. 2011;80:294–303.