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Chemical Structure : Takeda103A
CAS No.: 865609-72-9
Catalog No.: PC-38542Not For Human Use, Lab Use Only.
Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $148 | In stock | |
| 10 mg | $248 | In stock | |
| 25 mg | $448 | In stock | |
| 50 mg | $728 | In stock | |
| 100 mg | Get quote |
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Takeda103A is a potent, selective GRK2 inhibitor with IC50 of 0.02 uM, 450-fold selectivity over GRK5.
| M.Wt | 463.49 | |
| Formula | C24H23F2N7O | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
N-[(2,6-Difluorophenyl)methyl]-3-[[[4-propyl-5-(4-pyrimidinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-benzamide |
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1. Helen V Waldschmidt, et al. J Med Chem. 2016 Apr 28;59(8):3793-807.
2. Thal DM, et al. Mol Pharmacol. 2011;80:294–303.
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